SCHEMBL20140304

SCHEMBL20140304

Cc1cccc(N2CCN(C(=O)c3cc(CN4CCCN(c5ccccc5C#N)CC4)ccc3C)CC2)n1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 7/20 0.44
MTOR P42345 3/20 0.44
RPTOR Q8N122 3/20 0.44
MLST8 Q9BVC4 3/20 0.44
PARP1 P09874 1/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 2/20 0.40
DRD4 P21917 2/20 0.40
PHGDH O43175 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
DRD2 P14416 1/20 0.40
HTR2A P28223 1/20 0.40
DRD3 P35462 1/20 0.40
THPO P40225 1/20 0.40
HIF1A Q16665 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20156963 0.98 GBA1 (0.45) GBA1MTORRPTORMLST8PARP1
SCHEMBL20141546 0.87 MTOR (0.47) GBA1MTORRPTORMLST8MEN1
SCHEMBL20140044 0.87 MTOR (0.54) MTORRPTORMLST8PARP1MEN1
SCHEMBL20156808 0.86 MTOR (0.38) GBA1MTORRPTORMLST8PARP1
SCHEMBL20140777 0.85 DRD4 (0.43) GBA1MTORRPTORMLST8MEN1
SCHEMBL20157539 0.85 MTOR (0.46) MTORRPTORMLST8PARP1MEN1
SCHEMBL20140693 0.85 HCRTR1 (0.49) GBA1MTORRPTORMLST8PARP1
SCHEMBL20157255 0.85 MTOR (0.40) GBA1MTORRPTORMLST8PARP1
SCHEMBL20141182 0.85 PARP1 (0.48) MTORRPTORMLST8PARP1KDM4E
SCHEMBL20140897 0.85 MTOR (0.45) GBA1MTORRPTORMLST8PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089433-A1 PHENYL mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed
WO-2018089433-A1 PHENYL mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed