SCHEMBL20140692

SCHEMBL20140692

CNC(=O)c1ccccc1N1CCN(C(=O)O)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
RBP4 P02753 3/20 0.44
ALDH1A1 P00352 5/20 0.44
MYC P01106 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
KMT2A Q03164 2/20 0.44
MEN1 O00255 1/20 0.44
USP2 O75604 1/20 0.44
AR P10275 1/20 0.44
GAA P10253 1/20 0.44
NPC1 O15118 1/20 0.43
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
HTR1A P08908 1/20 0.42
DRD2 P14416 1/20 0.42
HTR2A P28223 1/20 0.42
KDM4E B2RXH2 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29496346 0.84 NPC1 (0.56) TSHRSMN1; SMN2ALDH1A1NPSR1KMT2A
SCHEMBL6262435 0.83 DRD2 (0.54) NPSR1HTR1ADRD2HTR2A
SCHEMBL21360304 0.82 BACE1 (0.54) SMN1; SMN2ALDH1A1NPSR1KMT2AMEN1
SCHEMBL20141942 0.80 MTOR (0.49) TSHRSMN1; SMN2ALDH1A1KMT2AMEN1
SCHEMBL1742847 0.80 ADRB1 (0.51) TSHRGAACYP2C19CYP1A2HTR1A
SCHEMBL10153998 0.80 ALDH1A1 (0.51) TSHRSMN1; SMN2ALDH1A1KMT2AMEN1
SCHEMBL6826072 0.79 ALDH1A1 (0.52) SMN1; SMN2ALDH1A1NPSR1KMT2AMEN1
SCHEMBL631024 0.76 AKR1C3 (0.65) TSHRALDH1A1MYCKMT2AAR
SCHEMBL20140930 0.75 GAA (0.38) TSHRSMN1; SMN2GAAHTR1ADRD2
SCHEMBL418681 0.75 RBP4 (0.46) TSHRSMN1; SMN2RBP4ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538091-A1 PHENYL AMINO PIPERIDINE mTORC INHIBITORS AND USES THEREOF Navitor Pharmaceuticals, Inc. (US) 2019-09-18 EP disclosed
WO-2018089433-A1 PHENYL mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed
WO-2018089499-A1 PHENYL AMINO PIPERIDINE mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed