SCHEMBL20141073

SCHEMBL20141073

CS(=O)(=NC(=O)O)c1c(F)cccc1F

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PKM P14618 4/20 0.39
PKLR P30613 1/20 0.39
KEAP1 Q14145 1/20 0.39
CES2 O00748 2/20 0.38
CES1 P23141 2/20 0.38
HTT P42858 1/20 0.37
ALB P02768 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
TDP1 Q9NUW8 1/20 0.35
SLC9A1 P19634 1/20 0.35
BCHE P06276 1/20 0.34
TTR P02766 1/20 0.34
PTGS2 P35354 1/20 0.34
ALOX15 P16050 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20129702 0.77 PKM (0.37) PKMPKLRHTT
SCHEMBL4139118 0.71 PKM (0.50) PKMPKLRKEAP1CES2CES1
SCHEMBL31046855 0.70 ALB (0.53) PKMPKLRKEAP1CES2CES1
SCHEMBL2576801 0.70 ALB (0.53) PKMPKLRKEAP1CES2CES1
SCHEMBL22693287 0.69 STS (0.45) PKMPKLRHTTSMN1; SMN2
SCHEMBL25388212 0.68 L3MBTL1 (0.38) PKMTDP1PTGS2ALOX15
SCHEMBL13784495 0.68 KMT2A (0.45)
SCHEMBL25387889 0.67 ALDH1A1 (0.53) PKMPKLRTDP1
SCHEMBL14676121 0.67 HSD11B1 (0.47) PKMPKLRKEAP1SMN1; SMN2ALOX15
SCHEMBL25386498 0.67 ALDH1A1 (0.53) PKMPKLRTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538091-A1 PHENYL AMINO PIPERIDINE mTORC INHIBITORS AND USES THEREOF Navitor Pharmaceuticals, Inc. (US) 2019-09-18 EP disclosed
WO-2018089499-A1 PHENYL AMINO PIPERIDINE mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed