SCHEMBL20142913

SCHEMBL20142913

CCN1N=C(c2ccc(Br)cc2)CC(C)(C)C1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
GAA P10253 5/20 0.38
NR1H2 P55055 1/20 0.36
NR1H3 Q13133 1/20 0.36
L3MBTL1 Q9Y468 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
FPR1 P21462 2/20 0.34
FPR2 P25090 2/20 0.34
LMNA P02545 4/20 0.33
MAPT P10636 3/20 0.33
KDM4E B2RXH2 2/20 0.33
PDE4B Q07343 2/20 0.33
ALDH1A1 P00352 2/20 0.33
CNR1 P21554 1/20 0.33
PAX8 Q06710 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
ADORA2A P29274 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20138839 0.86 CYP19A1 (0.39) SMN1; SMN2NPC1RAB9AL3MBTL1MEN1
SCHEMBL20138970 0.85 FPR1 (0.37) SMN1; SMN2NPC1RAB9AGAAL3MBTL1
SCHEMBL20159360 0.84 NPC1 (0.44) SMN1; SMN2NPC1RAB9AGAAL3MBTL1
SCHEMBL20159374 0.84 SMN1; SMN2 (0.39) SMN1; SMN2NPC1RAB9AGAAL3MBTL1
SCHEMBL20138895 0.83 SMN1; SMN2 (0.43) SMN1; SMN2NPC1RAB9AGAAMEN1
SCHEMBL20159737 0.81 RAB9A (0.36) SMN1; SMN2NPC1RAB9AGAAL3MBTL1
SCHEMBL20159532 0.81 SMN1; SMN2 (0.41) SMN1; SMN2NPC1RAB9AGAAMEN1
SCHEMBL20142960 0.81 SMN1; SMN2 (0.41) SMN1; SMN2NPC1RAB9AGAAL3MBTL1
SCHEMBL20159747 0.79 GSK3B (0.40) SMN1; SMN2RAB9AGAAMEN1KMT2A
SCHEMBL20138995 0.76 PDE4A (0.45) SMN1; SMN2NPC1RAB9AGAAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086703-A1 DIHYDROPYRIDAZINONES SUBSTITUTED WITH PHENYLUREAS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-05-17 WO disclosed
WO-2018086703-A1 DIHYDROPYRIDAZINONES SUBSTITUTED WITH PHENYLUREAS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-05-17 WO disclosed