SCHEMBL20145210

SCHEMBL20145210

CN1CCC[C@@H](Nc2ncc(C(F)(F)F)cn2)C1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
IL1B P01584 11/20 0.49
NLRP3 Q96P20 5/20 0.47
KAT2B Q92831 5/20 0.45
BPTF Q12830 1/20 0.45
CDK7 P50613 1/20 0.45
CCNH P51946 1/20 0.45
MNAT1 P51948 1/20 0.45
TRPV1 Q8NER1 1/20 0.44
CCNT1 O60563 1/20 0.43
CCNK O75909 1/20 0.43
CCNE1 P24864 1/20 0.43
CDK2 P24941 1/20 0.43
CDK9 P50750 1/20 0.43
CDK12 Q9NYV4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20145261 0.83 IL1B (0.55) IL1BNLRP3CCNKCDK2CDK12
SCHEMBL20144869 0.83 IL1B (0.55) IL1BNLRP3CCNKCDK2CDK12
SCHEMBL24968865 0.82 IDH2 (0.54) CCNKCCNE1CDK2CDK12
SCHEMBL25596437 0.81 CDK7 (0.52) IL1BNLRP3CDK7CCNHMNAT1
SCHEMBL20144776 0.81 IL1B (0.53) IL1BNLRP3KAT2BBPTF
SCHEMBL18607391 0.80 ULK1 (0.55)
SCHEMBL15951534 0.80 CDK7 (0.51) IL1BNLRP3KAT2BBPTFCDK7
SCHEMBL11989612 0.78 HRH4 (0.45) IL1BNLRP3KAT2BBPTFCCNT1
SCHEMBL25226590 0.78 MAPK3 (0.50) CCNKCDK12
SCHEMBL16187048 0.77 IL1B (0.53) IL1BNLRP3TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970207-B1 SUBSTITUTED PIPERIDINE COMPOUNDS AND THEIR USE AS OREXIN RECEPTOR MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2018-05-16 EP disclosed