SCHEMBL2014653

SCHEMBL2014653

OCCc1cc(Cl)c2ccncc2c1-c1cccc(F)c1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CSNK2A2 P19784 2/20 0.39
CSNK2B P67870 1/20 0.39
CYP17A1 P05093 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
DGAT2 Q96PD7 4/20 0.36
NT5E P21589 1/20 0.35
ADORA1 P30542 1/20 0.34
RPS6KA3 P51812 1/20 0.34
SLC22A12 Q96S37 1/20 0.34
HPGDS O60760 1/20 0.33
GCGR P47871 1/20 0.33
GRM5 P41594 1/20 0.33
DPP4 P27487 1/20 0.33
FYN P06241 1/20 0.33
IDO1 P14902 1/20 0.33
CSNK2A1 P68400 1/20 0.32
MAPK14 Q16539 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2015154 0.88 TAAR1 (0.41) CSNK2A2CSNK2BCYP17A1CYP3A4CYP11B1
SCHEMBL2017932 0.81 SLC22A12 (0.40) CSNK2A2CSNK2BCYP17A1CYP3A4CYP11B1
SCHEMBL2019261 0.80 PIK3CD (0.44) CYP17A1CYP3A4CYP11B1CYP11B2NT5E
SCHEMBL2014651 0.76 PIK3CD (0.39) CSNK2A2CSNK2BCYP17A1CYP3A4CYP11B1
SCHEMBL2015153 0.74 BCL2 (0.41) CSNK2A2CSNK2BCYP17A1CYP3A4CYP11B1
SCHEMBL2012666 0.72 TAAR1 (0.47) NT5E
SCHEMBL15621376 0.71 PIK3CD (0.38) CSNK2A2CSNK2BCYP17A1CYP3A4CYP11B1
SCHEMBL12470054 0.71 PIK3CD (0.38) CSNK2A2CSNK2BCYP17A1CYP3A4CYP11B1
SCHEMBL2016661 0.70 PIK3CD (0.36) CYP17A1CYP3A4CYP11B1CYP11B2ADORA1
SCHEMBL15617723 0.69 BCL2 (0.38) CSNK2A2CSNK2BCYP17A1CYP3A4CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011075630-A1 SUBSTITUTED FUSED ARYL AND HETEROARYL DERIVATIVES AS PI3K INHIBITORS INCYTE CORPORATION (US) 2011-06-23 WO disclosed