SCHEMBL2015154

SCHEMBL2015154

NCCc1cc(Cl)c2ccncc2c1-c1cccc(F)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 6/20 0.41
HTR6 P50406 2/20 0.36
CYP17A1 P05093 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
CSNK2A2 P19784 1/20 0.36
CSNK2B P67870 1/20 0.36
NT5E P21589 1/20 0.35
MGAT2 Q10469 1/20 0.35
DPP4 P27487 1/20 0.35
DGAT2 Q96PD7 3/20 0.34
CSNK1A1 P48729 1/20 0.34
CSNK1D P48730 1/20 0.34
CSNK1E P49674 1/20 0.34
CSNK1G2 P78368 1/20 0.34
CSNK1G1 Q9HCP0 1/20 0.34
SLC22A12 Q96S37 1/20 0.34
LOXL2 Q9Y4K0 1/20 0.33
CCNT1 O60563 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2014653 0.88 CSNK2A2 (0.39) CYP17A1CYP3A4CYP11B1CYP11B2CSNK2A2
SCHEMBL2012666 0.85 TAAR1 (0.47) TAAR1NT5E
SCHEMBL2017932 0.81 SLC22A12 (0.40) CYP17A1CYP3A4CYP11B1CYP11B2CSNK2A2
SCHEMBL12491178 0.80 BCL2 (0.47) TAAR1CYP17A1CYP3A4CYP11B1CYP11B2
SCHEMBL2015779 0.79 PIK3CD (0.44) TAAR1CYP3A4
SCHEMBL2017066 0.78 TAAR1 (0.43) TAAR1NT5EDPP4CCNT1CDK9
SCHEMBL2015153 0.76 BCL2 (0.41) CYP17A1CYP3A4CYP11B1CYP11B2CSNK2A2
SCHEMBL2014651 0.74 PIK3CD (0.39) CYP17A1CYP3A4CYP11B1CYP11B2CSNK2A2
Trifluoroacetic Acid SCHEMBL2012078 0.73 BCL2 (0.41) TAAR1CYP3A4NT5E
SCHEMBL12470054 0.71 PIK3CD (0.38) CYP17A1CYP3A4CYP11B1CYP11B2CSNK2A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011075630-A1 SUBSTITUTED FUSED ARYL AND HETEROARYL DERIVATIVES AS PI3K INHIBITORS INCYTE CORPORATION (US) 2011-06-23 WO disclosed