SCHEMBL20146789

SCHEMBL20146789

Cc1cc(-c2c[nH]/c(=N\C(C)N)cn2)ccc1C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CAMKK2 Q96RR4 3/20 0.43
LDHA P00338 3/20 0.41
NEK2 P51955 1/20 0.39
RXRB P28702 2/20 0.38
RXRA P19793 1/20 0.37
PIM1 P11309 1/20 0.37
CSNK2A1 P68400 1/20 0.37
LDHB P07195 2/20 0.36
GABRP O00591 1/20 0.36
GABRD O14764 1/20 0.36
GABRA1 P14867 1/20 0.36
GABRB1 P18505 1/20 0.36
GABRG2 P18507 1/20 0.36
GABRB3 P28472 1/20 0.36
GABRA5 P31644 1/20 0.36
GABRA3 P34903 1/20 0.36
GABRA2 P47869 1/20 0.36
GABRB2 P47870 1/20 0.36
GABRA4 P48169 1/20 0.36
GABRE P78334 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL481658 0.73 GABRP (0.55) CAMKK2LDHANEK2RXRBRXRA
SCHEMBL1498034 0.67 RXRB (0.70) CAMKK2LDHARXRBRXRARARB
SCHEMBL29771992 0.67 RXRB (0.70) CAMKK2LDHARXRBRXRARARB
SCHEMBL18191217 0.65 ALPL (0.55) CAMKK2LDHANEK2RXRBRXRA
Hydrochloric Acid SCHEMBL4365452 0.65 RXRB (0.68) CAMKK2LDHARXRBRXRARARB
Hydrochloric Acid SCHEMBL9150803 0.65 RXRB (0.68) CAMKK2LDHARXRBRXRARARB
SCHEMBL17177748 0.64 RXRB (0.71) CAMKK2LDHARXRBRXRARARB
SCHEMBL11517517 0.62 RXRB (0.51) CAMKK2LDHANEK2RXRBRXRA
SCHEMBL20768653 0.62 HSD17B10 (0.49) RXRBRXRAGABRPGABRDGABRA1
SCHEMBL21932509 0.62 HSD17B10 (0.49) RXRBRXRAGABRPGABRDGABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3321268-A1 BICYCLIC HETEROARYL DERIVATIVES AS MNK1 AND MNK2 MODULATORS AND USES THEREOF Agency For Science, Technology And Research (SG) 2018-05-16 EP disclosed