SCHEMBL20147149

SCHEMBL20147149

COc1ccc(C(O)n2c3ccc(OC)cc3c3ccncc32)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.46
MAOB P27338 1/20 0.46
HASPIN Q8TF76 1/20 0.43
CHUK O15111 1/20 0.42
ACHE P22303 4/20 0.40
KDM4E B2RXH2 4/20 0.40
MAPT P10636 4/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
BCHE P06276 2/20 0.40
HTT P42858 2/20 0.40
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40
HSD17B10 Q99714 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
ROCK2 O75116 3/20 0.39
CASR P41180 2/20 0.39
GRIN1 Q05586 1/20 0.39
GRIN2A Q12879 1/20 0.39
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12464508 0.83 MAOA (0.51) MAOAMAOBHASPINCHUKACHE
SCHEMBL20147143 0.80 DYRK1A (0.41) MAOAMAOBHASPINCHUKACHE
SCHEMBL4166593 0.76 HASPIN (0.52) MAOAMAOBHASPINCHUKACHE
SCHEMBL12464614 0.76 MAPT (0.64) MAOAMAOBHASPINCHUKACHE
SCHEMBL20135890 0.72 AKR1C3 (0.53) KDM4EMAPTMEN1KMT2ACYP1A2
SCHEMBL12464506 0.70 MAOA (0.49) MAOAMAOBHASPINCHUKACHE
SCHEMBL24277027 0.69 MAOA (0.48) MAOAMAOBHASPINCHUKACHE
SCHEMBL20135910 0.68 LMNA (0.56) ACHEKDM4EMAPTMEN1KMT2A
SCHEMBL1921708 0.68 HASPIN (0.61) MAOAMAOBHASPINCHUKACHE
SCHEMBL4176158 0.68 HASPIN (0.48) MAOAMAOBHASPINCHUKACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3321264-A1 SELECTIVE INHIBITORS OF GENOTOXIC STRESS-INDUCED IKK/NF-KB PATHWAYS Max-Delbrück-Centrum für Molekulare Medizin in der Helmholtz-Gemeinschaft (DE) 2018-05-16 EP disclosed