SCHEMBL2014823

SCHEMBL2014823

CCn1c(CNC(=O)c2nc(Cl)c(N)nc2N)nc2ccc(O)cc21

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.45
RPS6KA5 O75582 1/20 0.43
SCNN1A P37088 6/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
CTSA P10619 2/20 0.38
TP53 P04637 3/20 0.37
GRM5 P41594 1/20 0.36
LMNA P02545 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
TSHR P16473 1/20 0.36
THPO P40225 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2040435 0.91 HTT (0.45) HTTMEN1KMT2ACTSATP53
SCHEMBL2016331 0.90 HTT (0.52) HTTSCNN1AMEN1KMT2ACTSA
SCHEMBL2016153 0.89 HTT (0.44) HTTSCNN1AMEN1KMT2ACTSA
Iodide SCHEMBL2019625 0.88 HTT (0.43) HTTSCNN1AMEN1KMT2ACTSA
SCHEMBL2017836 0.88 HTT (0.46) HTTSCNN1AMEN1KMT2ATP53
SCHEMBL2020338 0.88 HTT (0.46) HTTRPS6KA5SCNN1AMEN1KMT2A
SCHEMBL16408252 0.88 RPS6KA5 (0.43) HTTRPS6KA5SCNN1ATP53
SCHEMBL2015344 0.87 HTT (0.47) HTTMEN1KMT2ACTSATP53
SCHEMBL12635756 0.87 HTT (0.49) HTTMEN1KMT2ATSHR
SCHEMBL2018438 0.87 SCNN1A (0.44) HTTSCNN1ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3022198-B1 NOVEL 5-SUBSTITUTED BENZIMIDAZOLIUM COMPOUNDS BOEHRINGER INGELHEIM INT (DE) 2019-09-11 EP disclosed
EP-3022197-B1 NOVEL TETRA- AND PENTASUBSTITUTED BENZIMIDAZOLIUM COMPOUNDS BOEHRINGER INGELHEIM INT (DE) 2017-09-06 EP disclosed
US-9073954-B2 5-substituted benzimidazolium compounds BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2015-07-07 US disclosed
US-9073954-B2 5-substituted benzimidazolium compounds BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2015-07-07 US disclosed
WO-2015007516-A1 NOVEL 5-SUBSTITUTED BENZIMIDAZOLIUM COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2015-01-22 WO disclosed
WO-2011079087-A1 ENAC BLOCKERS GLAXO GROUP LIMITED (GB) 2011-06-30 WO disclosed
WO-2011079087-A1 ENAC BLOCKERS GLAXO GROUP LIMITED (GB) 2011-06-30 WO disclosed