SCHEMBL2020338

SCHEMBL2020338

CCn1c(CNC(=O)c2nc(Cl)c(N)nc2N)nc2ccc(CO)cc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.46
S1PR1 P21453 1/20 0.44
SCNN1A P37088 3/20 0.41
CYP1A2 P05177 2/20 0.39
CYP2D6 P10635 2/20 0.39
THPO P40225 2/20 0.39
HSD17B10 Q99714 2/20 0.39
TP53 P04637 1/20 0.39
CYP3A4 P08684 1/20 0.39
TSHR P16473 1/20 0.39
KMT2A Q03164 2/20 0.39
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 2/20 0.39
GLA P06280 2/20 0.39
HPGD P15428 2/20 0.39
GMNN O75496 1/20 0.39
LMNA P02545 1/20 0.39
MAPK1 P28482 1/20 0.39
PMP22 Q01453 1/20 0.39
ACSS2 Q9NR19 6/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2040435 0.89 HTT (0.45) HTTCYP1A2CYP2D6THPOHSD17B10
SCHEMBL2014255 0.89 HTT (0.41) HTTSCNN1ACYP1A2CYP2D6THPO
SCHEMBL2016331 0.88 HTT (0.52) HTTSCNN1ACYP1A2CYP2D6THPO
SCHEMBL2014823 0.88 HTT (0.45) HTTSCNN1ACYP1A2CYP2D6THPO
SCHEMBL2018304 0.87 HTT (0.40) HTTSCNN1ACYP1A2CYP2D6THPO
SCHEMBL2016749 0.87 ACSS2 (0.41) HTTSCNN1ACYP1A2CYP2D6THPO
SCHEMBL2016153 0.87 HTT (0.44) HTTSCNN1ACYP1A2CYP2D6THPO
SCHEMBL2018137 0.87 ACSS2 (0.39) HTTSCNN1ACYP1A2CYP2D6THPO
SCHEMBL2014097 0.87 HTT (0.39) HTTSCNN1ACYP1A2CYP2D6THPO
Iodide SCHEMBL2019625 0.86 HTT (0.43) HTTSCNN1ACYP1A2CYP2D6THPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011079087-A1 ENAC BLOCKERS GLAXO GROUP LIMITED (GB) 2011-06-30 WO disclosed
WO-2011079087-A1 ENAC BLOCKERS GLAXO GROUP LIMITED (GB) 2011-06-30 WO disclosed