SCHEMBL2016331

SCHEMBL2016331

CCn1c(CNC(=O)c2nc(Cl)c(N)nc2N)nc2ccc(C)cc21

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.52
MAPT P10636 2/20 0.41
CTSA P10619 2/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
TLR8 Q9NR97 1/20 0.38
ACSS2 Q9NR19 1/20 0.38
TP53 P04637 4/20 0.37
GRM5 P41594 1/20 0.36
LMNA P02545 1/20 0.36
CYP1A2 P05177 2/20 0.36
CYP2D6 P10635 2/20 0.36
THPO P40225 2/20 0.36
HSD17B10 Q99714 2/20 0.36
CYP3A4 P08684 1/20 0.36
TSHR P16473 1/20 0.36
SCNN1A P37088 3/20 0.36
KDM4E B2RXH2 1/20 0.36
NPC1 O15118 1/20 0.36
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2015344 0.93 HTT (0.47) HTTMAPTCTSAMEN1KMT2A
SCHEMBL2040435 0.91 HTT (0.45) HTTMAPTCTSAMEN1KMT2A
SCHEMBL2014823 0.90 HTT (0.45) HTTCTSAMEN1KMT2ATP53
SCHEMBL2016153 0.89 HTT (0.44) HTTMAPTCTSAMEN1KMT2A
SCHEMBL2017836 0.88 HTT (0.46) HTTMEN1KMT2AACSS2TP53
Iodide SCHEMBL2019625 0.88 HTT (0.43) HTTMAPTCTSAMEN1KMT2A
SCHEMBL2020338 0.88 HTT (0.46) HTTMAPTCTSAMEN1KMT2A
SCHEMBL12635756 0.87 HTT (0.49) HTTMEN1KMT2AACSS2TSHR
SCHEMBL2018438 0.87 SCNN1A (0.44) HTTMAPTACSS2TP53SCNN1A
SCHEMBL2021620 0.87 HTT (0.45) HTTMAPTMEN1KMT2AACSS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011079087-A1 ENAC BLOCKERS GLAXO GROUP LIMITED (GB) 2011-06-30 WO disclosed
WO-2011079087-A1 ENAC BLOCKERS GLAXO GROUP LIMITED (GB) 2011-06-30 WO disclosed