SCHEMBL20148958

SCHEMBL20148958

Brc1ccc(C2CCN(Cc3ccccc3)C2)cc1

nearest known ligand 0.63

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ACHE P22303 4/20 0.60
BCHE P06276 3/20 0.60
BACE1 P56817 3/20 0.60
RORC P51449 2/20 0.56
MEN1 O00255 1/20 0.55
KMT2A Q03164 1/20 0.55
CCR5 P51681 1/20 0.53
SLC18A3 Q16572 2/20 0.52
SIGMAR1 Q99720 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4476807 0.94 MEN1 (0.63) ACHEBCHEBACE1MEN1KMT2A
SCHEMBL6701595 0.92 KMT2A (0.65) ACHEBCHEBACE1RORCMEN1
SCHEMBL22755777 0.89 MEN1 (0.68) ACHEBCHEBACE1MEN1KMT2A
SCHEMBL3598146 0.89 MEN1 (0.68) ACHEBCHEBACE1MEN1KMT2A
SCHEMBL6023725 0.89 MEN1 (0.68) ACHEBCHEBACE1MEN1KMT2A
SCHEMBL6902946 0.86 MEN1 (0.74) ACHEBCHEBACE1MEN1KMT2A
SCHEMBL4485265 0.85 CNR2 (0.60) ACHEBCHEBACE1MEN1KMT2A
SCHEMBL8844209 0.83 MEN1 (0.57) ACHEBCHEBACE1MEN1KMT2A
SCHEMBL6042732 0.82 RORC (0.58) ACHEBCHEBACE1RORCKMT2A
SCHEMBL31328443 0.82 CCR5 (0.49) ACHEBCHEBACE1RORCMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104860954-B A kind of phenyl ester spiropiperidines or spiropyrrolidines class compound and preparation method thereof 南京天印健华医药科技有限公司 2018-05-04 CN claimed
WO-2018089406-A1 ROR GAMMA MODULATORS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-17 WO disclosed
CN-104860954-B A kind of phenyl ester spiropiperidines or spiropyrrolidines class compound and preparation method thereof 南京天印健华医药科技有限公司 2018-05-04 CN disclosed