SCHEMBL20149045

SCHEMBL20149045

Fc1ccc(C2CNCC2c2ccc(-c3c(F)cccc3F)cc2)cc1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 5/20 0.40
SLC6A4 P31645 3/20 0.40
SLC6A3 Q01959 3/20 0.40
KDM1A O60341 2/20 0.40
NOS3 P29474 1/20 0.40
CHRNB2 P17787 1/20 0.40
CHRNA4 P43681 1/20 0.40
NOS1 P29475 1/20 0.40
NOS2 P35228 1/20 0.40
TTR P02766 1/20 0.40
ROCK2 O75116 2/20 0.38
RORC P51449 4/20 0.37
HTR2C P28335 2/20 0.37
HTR1A P08908 2/20 0.37
DRD1 P21728 1/20 0.37
HTR2A P28223 1/20 0.36
HTR2B P41595 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20149098 0.82 KDM1A (0.48) KDM1AROCK2HTR2CHTR1AHTR2A
SCHEMBL13615034 0.79 TTR (0.56) NOS1NOS2TTR
SCHEMBL23683586 0.76 RORC (0.56) TTRRORC
SCHEMBL20149049 0.76 RORC (0.56) TTRRORC
Hydrochloric Acid SCHEMBL23683617 0.75 RORC (0.55) TTRRORC
Hydrochloric Acid SCHEMBL23683618 0.75 RORC (0.55) TTRRORC
SCHEMBL20149028 0.74 KDM1A (0.45) SLC6A2SLC6A4SLC6A3KDM1AHTR2C
SCHEMBL20149036 0.74 KDM1A (0.45) SLC6A2SLC6A4SLC6A3KDM1AHTR2C
SCHEMBL23683613 0.72 RORC (0.59) RORCHTR2CHTR2A
SCHEMBL20139668 0.72 RORC (0.59) RORCHTR2CHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089406-A1 ROR GAMMA MODULATORS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-17 WO disclosed