SCHEMBL20149036

SCHEMBL20149036

Fc1ccc([C@H]2CNC[C@H]2c2ccc(Br)cc2)cc1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 7/20 0.45
KCNH2 Q12809 2/20 0.45
MAOB P27338 2/20 0.45
RCOR1 Q9UKL0 2/20 0.45
KDM1B Q8NB78 1/20 0.45
HTR2C P28335 5/20 0.40
HTR2B P41595 4/20 0.40
SLC6A2 P23975 2/20 0.40
HTR2A P28223 2/20 0.40
SLC6A4 P31645 2/20 0.40
SLC6A3 Q01959 2/20 0.40
TACR1 P25103 1/20 0.37
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20149028 1.00 KDM1A (0.45) KDM1AKCNH2MAOBRCOR1KDM1B
SCHEMBL20149098 0.77 KDM1A (0.48) KDM1AKCNH2MAOBHTR2CHTR2A
SCHEMBL2146401 0.76 KDM1A (0.45) KDM1AHTR2CHTR2BSLC6A2HTR2A
SCHEMBL16031353 0.76 KDM1A (0.45) KDM1AHTR2CHTR2BSLC6A2HTR2A
SCHEMBL16031350 0.76 KDM1A (0.45) KDM1AHTR2CHTR2BSLC6A2HTR2A
SCHEMBL2146399 0.76 KDM1A (0.45) KDM1AHTR2CHTR2BSLC6A2HTR2A
SCHEMBL7324342 0.74 QDPR (0.46) KDM1AKCNH2MAOBRCOR1KDM1B
SCHEMBL20148986 0.74 TACR1 (0.42) KDM1AKCNH2HTR2CHTR2BSLC6A2
SCHEMBL20149045 0.74 SLC6A2 (0.40) KDM1AHTR2CHTR2BSLC6A2HTR2A
SCHEMBL20139685 0.74 SLC6A3 (0.59) KCNH2SLC6A2SLC6A4SLC6A3TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089406-A1 ROR GAMMA MODULATORS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-17 WO disclosed