SCHEMBL20149104

SCHEMBL20149104

CC(=O)N1CCC(C(=O)N2CC(C)[C@H](c3ccc(-c4c(F)cccc4F)cc3)C2)CC1

nearest known ligand 0.71

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
RORC P51449 9/20 0.71
TACR1 P25103 9/20 0.47
TACR2 P21452 4/20 0.47
TACR3 P29371 2/20 0.47
PAX8 Q06710 1/20 0.43
TAC3 Q9UHF0 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23713149 0.83 RORC (1.00) RORCTACR1TACR2TACR3CYP3A4
SCHEMBL23713009 0.75 RORC (1.00) RORC
SCHEMBL20149048 0.73 RORC (0.77) RORCTACR3
SCHEMBL20149105 0.69 RORC (1.00) RORC
SCHEMBL20002952 0.69 RORC (0.47) RORCPAX8
SCHEMBL20149050 0.69 RORC (0.84) RORCTACR1TACR2
SCHEMBL20149129 0.69 RORC (0.80) RORCTACR1TACR2CYP3A4CYP2D6
SCHEMBL23713056 0.69 RORC (1.00) RORCTACR1CYP3A4CYP2D6CYP2C9
SCHEMBL15751783 0.69 TACR1 (0.70) RORCTACR1TACR2TACR3TAC3
SCHEMBL17086647 0.68 TACR1 (0.46) RORCTACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089406-A1 ROR GAMMA MODULATORS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-17 WO disclosed