SCHEMBL20002952

SCHEMBL20002952

O=CC1CCC(C(=O)N2CCC(c3ccc(-c4c(F)cccc4F)cc3)C2)CC1

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
RORC P51449 4/20 0.47
PAX8 Q06710 3/20 0.44
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
ATM Q13315 1/20 0.40
MGLL Q99685 1/20 0.39
HSD11B1 P28845 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12447952 0.73 RAB9A (0.61) NPC1RAB9AATMHSD11B1
SCHEMBL12447336 0.69 CCR5 (0.61) NPC1RAB9AATMHSD11B1
SCHEMBL12447948 0.69 CCR5 (0.61) NPC1RAB9AATMHSD11B1
SCHEMBL20149104 0.69 RORC (0.71) RORCPAX8
SCHEMBL16785546 0.66 NPC1 (0.54) NPC1RAB9A
SCHEMBL11178698 0.66 ALDH1A1 (0.58) NPC1RAB9AATMHSD11B1
SCHEMBL12447717 0.65 NAMPT (0.57) NPC1RAB9AATM
SCHEMBL20148966 0.65 CCR5 (0.48)
SCHEMBL13097359 0.65 HPGD (0.56) HSD11B1
SCHEMBL19988362 0.64 HTR2B (0.64) NPC1RAB9AATMHSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed