SCHEMBL20150284

SCHEMBL20150284

CNc1nc(N)ncc1Br

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
JAK1 P23458 1/20 0.46
TYK2 P29597 1/20 0.46
NUDT1 P36639 2/20 0.40
PTPN1 P18031 1/20 0.39
GRM4 Q14833 1/20 0.39
CHUK O15111 1/20 0.37
PDPK1 O15530 1/20 0.36
BCL6 P41182 2/20 0.36
IKBKE Q14164 1/20 0.35
TBK1 Q9UHD2 1/20 0.35
LRRK2 Q5S007 1/20 0.34
IGF1R P08069 1/20 0.33
DHFR P00374 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16011451 0.78 NUDT1 (0.42) JAK1TYK2NUDT1CHUKPDPK1
SCHEMBL24457928 0.78 FGFR1 (0.47)
SCHEMBL2745753 0.77 NUDT1 (0.58) NUDT1PTPN1GRM4BCL6DHFR
SCHEMBL2744648 0.75 BCL6 (0.56) TYK2NUDT1PTPN1CHUKPDPK1
SCHEMBL20150368 0.75 NUDT1 (0.40) NUDT1CHUKBCL6L3MBTL1
SCHEMBL14994344 0.75 BCL6 (0.56) NUDT1PTPN1GRM4BCL6LRRK2
SCHEMBL3139282 0.75 KMT2A (0.49) PDPK1LRRK2IGF1RL3MBTL1
SCHEMBL2745948 0.73 DHFR (0.43) NUDT1DHFR
SCHEMBL31403281 0.73 JAK1 (0.65) JAK1TYK2GRM4CHUKIGF1R
SCHEMBL13488651 0.72 PDE10A (0.43) JAK1TYK2NUDT1TBK1LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230295144-A1 2-polysubstituted aromatic ring-pyrimidine derivatives, preparation and medical application thereof UNIV ZHEJIANG (CN) 2023-09-21 US claimed
US-20210284625-A1 2-polysubstituted aromatic ring-pyrimidine derivatives, preparation and medical application thereof UNIV ZHEJIANG (CN) 2021-09-16 US claimed
EP-3530657-A1 2-POLYSUBSTITUTED AROMATIC RING-PYRIMIDINE DERIVATIVE AND PREPARATION AND MEDICAL USE Zhejiang University (CN) 2019-08-28 EP claimed
EP-4526318-A1 FLEX-NUCLEOSIDE ANALOGUES, NOVEL THERAPEUTICS AGAINST VIRUSES University of Maryland, Baltimore County (US) 2025-03-26 EP disclosed
US-20250092080-A1 FLEX-NUCLEOSIDE ANALOGUES, NOVEL THERAPEUTICS AGAINST VIRUSES UNIVERSITY OF MARYLAND, BALTIMORE COUNTY 2025-03-20 US disclosed
WO-2023225042-A1 FLEX-NUCLEOSIDE ANALOGUES, NOVEL THERAPEUTICS AGAINST VIRUSES UNIVERSITY OF MARYLAND, BALTIMORE COUNTY (US) 2023-11-23 WO disclosed
US-20230295144-A1 2-polysubstituted aromatic ring-pyrimidine derivatives, preparation and medical application thereof UNIV ZHEJIANG (CN) 2023-09-21 US disclosed
US-20230295144-A1 2-polysubstituted aromatic ring-pyrimidine derivatives, preparation and medical application thereof UNIV ZHEJIANG (CN) 2023-09-21 US disclosed
US-11591325-B2 2-polysubstituted aromatic ring-pyrimidine derivatives, preparation and medical application thereof ZHEJIANG UNIVERSITY (CN) 2023-02-28 US disclosed
US-11591325-B2 2-polysubstituted aromatic ring-pyrimidine derivatives, preparation and medical application thereof ZHEJIANG UNIVERSITY (CN) 2023-02-28 US disclosed
US-20210284625-A1 2-polysubstituted aromatic ring-pyrimidine derivatives, preparation and medical application thereof UNIV ZHEJIANG (CN) 2021-09-16 US disclosed
US-20210284625-A1 2-polysubstituted aromatic ring-pyrimidine derivatives, preparation and medical application thereof UNIV ZHEJIANG (CN) 2021-09-16 US disclosed
EP-3530657-A1 2-POLYSUBSTITUTED AROMATIC RING-PYRIMIDINE DERIVATIVE AND PREPARATION AND MEDICAL USE Zhejiang University (CN) 2019-08-28 EP disclosed
EP-3530657-A1 2-POLYSUBSTITUTED AROMATIC RING-PYRIMIDINE DERIVATIVE AND PREPARATION AND MEDICAL USE Zhejiang University (CN) 2019-08-28 EP disclosed
WO-2018086546-A1 2-POLYSUBSTITUTED AROMATIC RING-PYRIMIDINE DERIVATIVE AND PREPARATION AND MEDICAL USE 浙江大学 2018-05-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11591325-B2 2-polysubstituted aromatic ring-pyrimidine derivatives, preparation and medical application thereof CHEK1, PLK1, CHEK2 JAK1 193/4885TYK2 393/4885NUDT1 665/4885
US-20250092080-A1 FLEX-NUCLEOSIDE ANALOGUES, NOVEL THERAPEUTICS AGAINST VIRUSES FLNA, PNP, SMCHD1 JAK1 2837/4885TYK2 470/4885NUDT1 65/4885
US-20230295144-A1 2-polysubstituted aromatic ring-pyrimidine derivatives, preparation and medical application thereof CHEK1, PLK1, CHEK2 JAK1 193/4885TYK2 393/4885NUDT1 665/4885
US-20210284625-A1 2-polysubstituted aromatic ring-pyrimidine derivatives, preparation and medical application thereof CHEK1, PLK1, CHEK2 JAK1 193/4885TYK2 393/4885NUDT1 665/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.