SCHEMBL2013705

SCHEMBL2013705

Fc1cc(F)cc(-c2[c]ccc(C(F)(F)F)c2)c1

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
RXRA P19793 1/20 0.33
RXRB P28702 1/20 0.33
RXRG P48443 1/20 0.33
PDE2A O00408 2/20 0.32
CES2 O00748 1/20 0.32
TSHR P16473 1/20 0.31
MAPK1 P28482 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1690372 0.85 SMN1; SMN2 (0.34) PDE2ACES2MAPK1
SCHEMBL2431003 0.84 PTPN1 (0.39) CES2TSHRMAPK1
SCHEMBL8078153 0.81 KIF11 (0.43) CES2TSHR
SCHEMBL2296580 0.80 RAPGEF4 (0.35) PDE2ACES2TSHRMAPK1
SCHEMBL1370057 0.79 KIF11 (0.47) CES2TSHRMAPK1
SCHEMBL2015248 0.79 TRPA1 (0.43) PDE2A
SCHEMBL4453497 0.78 NOTUM (0.32)
SCHEMBL2204411 0.78 NOTUM (0.43) CES2TSHRMAPK1
SCHEMBL2013527 0.77 GABRP (0.30)
SCHEMBL10340202 0.76 PTGDR2 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013182433-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2013-12-12 WO disclosed
EP-2547687-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2013-01-23 EP disclosed
EP-2513067-A1 METHOD FOR PRODUCING TRIAZOLINTHIONE DERIVATIVES AND INTERMEDIATES THEREOF BASF SE (DE) 2012-10-24 EP disclosed
WO-2011113820-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2011-09-22 WO disclosed
WO-2011073145-A1 METHOD FOR PRODUCING TRIAZOLINTHIONE DERIVATIVES AND INTERMEDIATES THEREOF BASF SE (DE) 2011-06-23 WO disclosed