SCHEMBL20153798

SCHEMBL20153798

N=Cc1cc(OCCc2ccc3c(n2)NCCC3)ccc1N

nearest known ligand 0.52

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 20/20 0.52
ITGAV P06756 20/20 0.52
ITGB6 P18564 7/20 0.50
ITGB5 P18084 5/20 0.50
ITGB1 P05556 1/20 0.50
ITGA2B P08514 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22600425 0.79 ITGB3 (0.46) ITGB3ITGAVITGB6ITGB5ITGB1
SCHEMBL860659 0.76 ITGB3 (0.56) ITGB3ITGAVITGB6ITGB5ITGB1
SCHEMBL29936679 0.75 ITGB3 (0.55) ITGB3ITGAVITGB6ITGB5ITGB1
SCHEMBL20139335 0.75 ITGB3 (0.55) ITGB3ITGAVITGB6ITGB5ITGB1
SCHEMBL22600427 0.75 ITGB3 (0.51) ITGB3ITGAVITGB6ITGB5ITGA2B
SCHEMBL23677919 0.71 ITGAV (0.60) ITGB3ITGAVITGB6ITGB5ITGB1
SCHEMBL21784941 0.71 ITGAV (0.54) ITGB3ITGAVITGB6ITGB5ITGB1
SCHEMBL4786884 0.71 ITGB3 (0.71) ITGB3ITGAVITGB6ITGB5ITGB1
SCHEMBL1815095 0.69 ITGAV (0.51) ITGB3ITGAVITGB6ITGB5ITGB1
SCHEMBL20021718 0.69 ITGB3 (0.56) ITGB3ITGAVITGB6ITGB5ITGB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089357-A1 INDAZOLE DERIVATIVES AS αV INTEGRIN ANTAGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-17 WO disclosed