SCHEMBL20155003

SCHEMBL20155003

Cn1cc2c(=O)n(C)cc(Br)c2n1

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 10/20 0.36
ADORA2A P29274 1/20 0.33
ADORA1 P30542 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
MAT2A P31153 4/20 0.32
NPSR1 Q6W5P4 1/20 0.31
BRD9 Q9H8M2 1/20 0.31
BRD7 Q9NPI1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20155066 0.87 MAT2A (0.34) BRD4ADORA2AADORA1MAT2ANPSR1
SCHEMBL20155470 0.79 BRD4 (0.35) BRD4ADORA2AADORA1L3MBTL1MAT2A
SCHEMBL20155118 0.79 NPC1 (0.40) BRD4MAT2A
SCHEMBL20154966 0.79 BRD4 (0.35) BRD4BRD9BRD7
SCHEMBL20155332 0.79 ADORA2A (0.36) BRD4ADORA2AADORA1MAT2A
SCHEMBL30975393 0.78
SCHEMBL20155436 0.76 TLR8 (0.41) BRD4
SCHEMBL20155089 0.75 PSMB5 (0.31) BRD4L3MBTL1
SCHEMBL20155605 0.75
SCHEMBL20155133 0.74 ADORA2A (0.37) ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112300154-B Nitrogen-containing heterocyclic compound, preparation method and application thereof 上海弘翊生物科技有限公司 2023-01-24 CN disclosed
CN-112300154-A Nitrogen-containing heterocyclic compound, preparation method and application thereof 上海弘翊生物科技有限公司 2021-02-02 CN disclosed
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed