SCHEMBL20155089

SCHEMBL20155089

CC(C)On1cc2c(=O)n(C)cc(Br)c2n1

nearest known ligand 0.31

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PSMB5 P28074 1/20 0.31
BRD4 O60885 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20154966 0.83 BRD4 (0.35) BRD4
SCHEMBL20155605 0.79
SCHEMBL20155332 0.76 ADORA2A (0.36) PSMB5BRD4
SCHEMBL20155003 0.75 BRD4 (0.36) BRD4L3MBTL1
SCHEMBL20155732 0.75 GSK3B (0.30)
SCHEMBL20155616 0.72 ALDH1A1 (0.38) BRD4
SCHEMBL20155118 0.70 NPC1 (0.40) BRD4
SCHEMBL20155045 0.69 ALDH1A1 (0.39) BRD4
SCHEMBL20155436 0.68 TLR8 (0.41) BRD4
SCHEMBL20155133 0.66 ADORA2A (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed