SCHEMBL20155332

SCHEMBL20155332

CC(C)n1cc2c(=O)n(C)cc(Br)c2n1

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.36
ADORA1 P30542 2/20 0.36
MAT2A P31153 1/20 0.34
BRD4 O60885 5/20 0.32
BRD2 P25440 2/20 0.32
BRD3 Q15059 2/20 0.32
CREBBP Q92793 2/20 0.32
LRRK2 Q5S007 2/20 0.32
PSMB5 P28074 1/20 0.30
AADAT Q8N5Z0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20155093 0.89 MAT2A (0.36) ADORA2AADORA1MAT2ABRD4BRD2
SCHEMBL20155003 0.79 BRD4 (0.36) ADORA2AADORA1MAT2ABRD4
SCHEMBL20155089 0.76 PSMB5 (0.31) BRD4PSMB5
SCHEMBL20154966 0.73 BRD4 (0.35) BRD4
SCHEMBL20155118 0.73 NPC1 (0.40) MAT2ABRD4
SCHEMBL20155436 0.71 TLR8 (0.41) BRD4BRD2BRD3CREBBP
SCHEMBL20155605 0.70
SCHEMBL20155133 0.69 ADORA2A (0.37) ADORA2A
SCHEMBL20155045 0.69 ALDH1A1 (0.39) BRD4LRRK2
SCHEMBL20155529 0.69 CNR2 (0.40) BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed