SCHEMBL20155043

SCHEMBL20155043

COCCn1cc2c(O)ncc(Br)c2n1

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 3/20 0.34
CYP1A2 P05177 1/20 0.32
MAP4K4 O95819 1/20 0.32
EGFR P00533 1/20 0.32
FRK P42685 1/20 0.32
MAPK9 P45984 1/20 0.32
CSNK1D P48730 1/20 0.32
SLK Q9H2G2 1/20 0.32
RECQL P46063 1/20 0.31
IRAK4 Q9NWZ3 2/20 0.31
HSD17B1 P14061 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20155691 0.80 NPC1 (0.40)
SCHEMBL20155391 0.75 LMNA (0.33)
SCHEMBL27192248 0.74 LRRK2 (0.36) LRRK2CYP1A2MAP4K4EGFRFRK
SCHEMBL20155045 0.72 ALDH1A1 (0.39) LRRK2CYP1A2
SCHEMBL20155044 0.72 MPO (0.38) LRRK2MAP4K4EGFRFRKMAPK9
SCHEMBL25105284 0.70 PTGER4 (0.38)
SCHEMBL23850448 0.70 ALDH1A1 (0.35) LRRK2CYP1A2MAP4K4EGFRFRK
SCHEMBL27077536 0.70 MAP4K4 (0.35) LRRK2CYP1A2MAP4K4EGFRFRK
SCHEMBL2596825 0.70 MAP4K4 (0.37) LRRK2CYP1A2MAP4K4EGFRFRK
SCHEMBL25105273 0.69 KDM4E (0.41) CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed