SCHEMBL20155045

SCHEMBL20155045

COCCn1cc2c(=O)n(C)cc(Br)c2n1

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 2/20 0.35
BRD4 O60885 7/20 0.35
RXFP1 Q9HBX9 1/20 0.33
LRRK2 Q5S007 3/20 0.33
KDM5B Q9UGL1 1/20 0.32
HSD17B10 Q99714 1/20 0.31
POLB P06746 1/20 0.30
PKM P14618 1/20 0.30
CYP1A2 P05177 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20155118 0.81 NPC1 (0.40) ALDH1A1KDM4EBRD4MEN1KMT2A
SCHEMBL20155529 0.79 CNR2 (0.40) ALDH1A1KDM4EBRD4POLBMEN1
SCHEMBL20154966 0.75 BRD4 (0.35) BRD4
SCHEMBL20155115 0.74 ADORA3 (0.50) ALDH1A1KDM4EBRD4CYP1A2MEN1
SCHEMBL20155003 0.74 BRD4 (0.36) BRD4
SCHEMBL20155043 0.72 LRRK2 (0.34) LRRK2CYP1A2
SCHEMBL20155605 0.72
SCHEMBL25105284 0.71 PTGER4 (0.38) ALDH1A1KMT2A
SCHEMBL20154927 0.71 MAT2A (0.40) ALDH1A1KDM4EMEN1KMT2A
SCHEMBL27077536 0.71 MAP4K4 (0.35) ALDH1A1KDM4ERXFP1LRRK2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed