SCHEMBL20155077

SCHEMBL20155077

CN(N)c1c(N)c(Br)cn(C)c1=O

nearest known ligand 0.30

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.30
TTK P33981 1/20 0.30
AURKB Q96GD4 1/20 0.30
INCENP Q9NQS7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20155558 0.87
SCHEMBL20155569 0.78 AURKA (0.34) AURKATTKAURKBINCENP
SCHEMBL15068063 0.71 AURKA (0.33) AURKATTKAURKBINCENP
SCHEMBL20155561 0.68 ALDH1A1 (0.40)
SCHEMBL16650601 0.63 BRD4 (0.34)
SCHEMBL20154923 0.60 BRD4 (0.38)
SCHEMBL106685 0.60 AURKA (0.49) AURKATTKAURKBINCENP
SCHEMBL23233752 0.59 BRD4 (0.38)
SCHEMBL16651641 0.59 BRD4 (0.58)
SCHEMBL22990247 0.59 MAP2K1 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed