SCHEMBL20155727

SCHEMBL20155727

CN1C=C(c2cc(N)ccc2Nc2ccc(Cl)cc2F)C(=N)C(=N)C1=O

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NUDT1 P36639 1/20 0.34
BRD4 O60885 2/20 0.33
TRPM5 Q9NZQ8 1/20 0.32
TAS2R14 Q9NYV8 1/20 0.31
TSHR P16473 1/20 0.31
MAPK14 Q16539 1/20 0.31
KDR P35968 4/20 0.30
FLT1 P17948 3/20 0.30
MAP2K1 Q02750 2/20 0.30
MAP2K2 P36507 1/20 0.30
KMT2A Q03164 2/20 0.30
EGFR P00533 2/20 0.30
FGFR1 P11362 1/20 0.30
PDGFRB P09619 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20155062 0.89 MAPK14 (0.39) BRD4TSHRMAPK14MAP2K1MAP2K2
SCHEMBL20155632 0.86 BPTF (0.37) BRD4KMT2A
SCHEMBL20155508 0.83 BRD4 (0.32) BRD4MAPK14
SCHEMBL20155138 0.77 MAPK14 (0.36) BRD4MAPK14KMT2A
SCHEMBL20155590 0.77 MAPK14 (0.36) BRD4MAPK14MAP2K1MAP2K2KMT2A
SCHEMBL20155748 0.75 MAPK14 (0.34) BRD4MAPK14KMT2A
SCHEMBL20155186 0.74 TDO2 (0.31)
SCHEMBL20155507 0.74 BRD4 (0.39) BRD4
SCHEMBL20155156 0.73 BPTF (0.33) BRD4KMT2A
SCHEMBL20155483 0.73 MAPK14 (0.37) BRD4MAPK14KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed