SCHEMBL20155156

SCHEMBL20155156

CN/C=C1\C(=N)C(c2cc(N)ccc2Nc2ccc(Cl)cc2)=CN(C)C1=O

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BPTF Q12830 1/20 0.33
BRD4 O60885 1/20 0.31
ALDH1A1 P00352 1/20 0.31
GAA P10253 1/20 0.31
ALOX15 P16050 1/20 0.31
HTT P42858 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20155632 0.87 BPTF (0.37) BPTFBRD4ALDH1A1GAAALOX15
SCHEMBL20155186 0.85 TDO2 (0.31)
SCHEMBL20155731 0.84
SCHEMBL20155590 0.82 MAPK14 (0.36) BRD4ALDH1A1MEN1KMT2A
SCHEMBL20155692 0.77 SLC6A2 (0.34) BRD4
SCHEMBL20155030 0.75 SCN9A (0.34)
SCHEMBL20155138 0.74 MAPK14 (0.36) BRD4ALDH1A1MEN1KMT2A
SCHEMBL20155146 0.74
SCHEMBL20155007 0.74 SLC6A2 (0.35) BRD4
SCHEMBL20155727 0.73 NUDT1 (0.34) BRD4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed