SCHEMBL20156942

SCHEMBL20156942

C[C@H]1CN(c2cccc3cc[nH]c23)CCN1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.40
LMNA P02545 2/20 0.40
HTR2C P28335 1/20 0.38
HRH4 Q9H3N8 1/20 0.37
PRKCQ Q04759 3/20 0.37
PRKCD Q05655 1/20 0.37
AHR P35869 1/20 0.37
HTR6 P50406 2/20 0.36
ADRB1 P08588 1/20 0.36
CYP2D6 P10635 2/20 0.36
NFKB1 P19838 2/20 0.36
HTR3E A5X5Y0 1/20 0.36
HTR3B O95264 1/20 0.36
CYP1A2 P05177 1/20 0.36
HTR1A P08908 1/20 0.36
NCF1 P14598 1/20 0.36
TSHR P16473 1/20 0.36
HTR1D P28221 1/20 0.36
HTR1B P28222 1/20 0.36
HTR2A P28223 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL20141711 0.88 HTR2C (0.39) ALDH1A1LMNAHTR2CHRH4PRKCQ
SCHEMBL3297385 0.79 HTR6 (0.57) ALDH1A1LMNAHTR2CHTR6ADRB1
SCHEMBL20141437 0.78 HTR1A (0.44) ALDH1A1LMNAHTR2CPRKCQPRKCD
SCHEMBL20141435 0.78 HTR1A (0.44) ALDH1A1LMNAHTR2CPRKCQPRKCD
SCHEMBL4244450 0.78 HTR6 (0.61) ALDH1A1LMNAHTR2CHRH4PRKCQ
SCHEMBL4247868 0.78 HTR6 (0.61) ALDH1A1LMNAHTR2CHRH4PRKCQ
SCHEMBL4244446 0.78 HTR6 (0.61) ALDH1A1LMNAHTR2CHRH4PRKCQ
SCHEMBL30146614 0.77 ADRB1 (0.64) HTR2CHTR6ADRB1HTR1AMAPT
SCHEMBL4247455 0.76 MKNK1 (0.39) ALDH1A1LMNAHTR2CPRKCQPRKCD
SCHEMBL4246453 0.76 MKNK1 (0.39) ALDH1A1LMNAHTR2CPRKCQPRKCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089433-A1 PHENYL mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed
WO-2018089493-A1 PYRROLE mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed