SCHEMBL20141437

SCHEMBL20141437

CC1CN(c2cccc3cn[nH]c23)CCN1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.44
ROCK2 O75116 3/20 0.43
ROCK1 Q13464 2/20 0.43
PRKCQ Q04759 4/20 0.42
PRKCD Q05655 2/20 0.42
NOS1 P29475 2/20 0.40
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
NFKB1 P19838 1/20 0.38
PRKD3 O94806 1/20 0.38
PRKCG P05129 1/20 0.38
PRKCB P05771 1/20 0.38
PRKCA P17252 1/20 0.38
PRKCH P24723 1/20 0.38
PRKCI P41743 1/20 0.38
PRKCE Q02156 1/20 0.38
PRKCZ Q05513 1/20 0.38
PRKD1 Q15139 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20141435 1.00 HTR1A (0.44) HTR1AROCK2ROCK1PRKCQPRKCD
SCHEMBL20140658 0.78 ROCK2 (0.50) ROCK2ROCK1PRKCQPRKCDPRKCI
SCHEMBL30146781 0.78 ROCK2 (0.43) ROCK2ROCK1PRKCQPRKCDNOS1
SCHEMBL20140662 0.78 ROCK2 (0.50) ROCK2ROCK1PRKCQPRKCDPRKCI
SCHEMBL20156942 0.78 ALDH1A1 (0.40) HTR1APRKCQPRKCDALDH1A1LMNA
SCHEMBL4247868 0.76 HTR6 (0.61) HTR1APRKCQPRKCDALDH1A1LMNA
SCHEMBL4244450 0.76 HTR6 (0.61) HTR1APRKCQPRKCDALDH1A1LMNA
SCHEMBL4244446 0.76 HTR6 (0.61) HTR1APRKCQPRKCDALDH1A1LMNA
SCHEMBL27630897 0.76 HTR1A (0.51) HTR1ANOS1CYP3A4PRKCZHTR2C
SCHEMBL20140653 0.75 PIM1 (0.41) ROCK2PRKCQPRKCDALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089433-A1 PHENYL mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed