SCHEMBL20157488

SCHEMBL20157488

COc1ccc(C(=O)c2ccc(C(C)Br)cc2Br)cc1F

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 5/20 0.49
LMNA P02545 4/20 0.49
MAPK1 P28482 2/20 0.49
RAB9A P51151 1/20 0.49
ALDH1A1 P00352 6/20 0.47
CYP11B1 P15538 1/20 0.43
CYP11B2 P19099 1/20 0.43
ACHE P22303 1/20 0.42
HPGD P15428 5/20 0.42
CYP1A2 P05177 2/20 0.42
CYP2C19 P33261 2/20 0.42
CYP2D6 P10635 1/20 0.42
TAS1R3 Q7RTX0 1/20 0.42
TAS1R1 Q7RTX1 1/20 0.42
CYP3A4 P08684 2/20 0.40
CYP2C9 P11712 1/20 0.40
TSHR P16473 1/20 0.40
KMT2A Q03164 2/20 0.40
MAPT P10636 5/20 0.39
NPSR1 Q6W5P4 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20158085 0.91 HTT (0.50) HTTLMNAMAPK1RAB9AALDH1A1
SCHEMBL21362792 0.84 ALDH1A1 (0.44) HTTALDH1A1HPGDCYP1A2CYP2C19
SCHEMBL21564711 0.83 ALDH1A1 (0.43) HTTMAPK1RAB9AALDH1A1HPGD
SCHEMBL20158084 0.82 HTT (0.54) HTTLMNAMAPK1RAB9AALDH1A1
SCHEMBL20157647 0.81 ALDH1A1 (0.44) HTTLMNAMAPK1RAB9AALDH1A1
SCHEMBL21362666 0.81 RAB9A (0.38) HTTLMNAMAPK1RAB9AALDH1A1
SCHEMBL16364815 0.80 HTT (0.58) HTTLMNAMAPK1RAB9AALDH1A1
SCHEMBL20157564 0.80 LMNA (0.42) HTTLMNAALDH1A1HPGDKMT2A
SCHEMBL20158040 0.79 ACHE (0.54) HTTLMNAMAPK1RAB9AALDH1A1
SCHEMBL9774382 0.77 LMNA (0.44) HTTLMNAMAPK1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086605-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed