SCHEMBL20157673

SCHEMBL20157673

C=C(c1ccc(F)cc1)c1cc(Cl)c(N)cc1Br

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA P19793 2/20 0.35
ALDH1A1 P00352 3/20 0.33
POLB P06746 2/20 0.33
HPGD P15428 2/20 0.33
MAOA P21397 2/20 0.33
MAOB P27338 2/20 0.33
GAA P10253 1/20 0.32
HDAC1 Q13547 1/20 0.32
HTR4 Q13639 1/20 0.31
CA12 O43570 2/20 0.30
CA1 P00915 2/20 0.30
CA2 P00918 2/20 0.30
CA9 Q16790 2/20 0.30
SLC9A1 P19634 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
KEAP1 Q14145 1/20 0.30
RARB P10826 1/20 0.30
RARG P13631 1/20 0.30
CA7 P43166 1/20 0.30
CA14 Q9ULX7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20157680 0.82 POLB (0.42) RXRAALDH1A1POLBHPGDHDAC1
SCHEMBL21362581 0.73 ANO1 (0.40) RXRAMAOBSMN1; SMN2
SCHEMBL21550431 0.72 HPGD (0.44) ALDH1A1POLBHPGDGAAKEAP1
SCHEMBL21362535 0.69 SMN1; SMN2 (0.43) RXRAALDH1A1HPGDCA12CA1
SCHEMBL10704841 0.69 FLT1 (0.47) ALDH1A1POLBHPGDHDAC1SMN1; SMN2
SCHEMBL20157693 0.69 MAPT (0.49) ALDH1A1POLB
SCHEMBL31619553 0.68 ALDH1A1 (0.46) ALDH1A1HPGDMAOAMAOBGAA
SCHEMBL10389925 0.68 HSD11B1 (0.46) ALDH1A1POLBHPGDSMN1; SMN2
SCHEMBL20244265 0.68 HSD11B1 (0.44) ALDH1A1POLBHPGDMAOAMAOB
SCHEMBL20157692 0.68 MAPK1 (0.44) RXRAALDH1A1POLBHPGDMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086605-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed