SCHEMBL20157893

SCHEMBL20157893

Cc1ccc(C(=O)c2ccc(C)cc2Br)c(F)c1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.41
MAPT P10636 2/20 0.41
MAPK1 P28482 1/20 0.41
HTT P42858 1/20 0.41
DGAT1 O75907 1/20 0.41
CSNK2A1 P68400 1/20 0.39
MYC P01106 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38
LOXL2 Q9Y4K0 1/20 0.38
CES2 O00748 1/20 0.37
CES1 P23141 1/20 0.37
CPS1 P31327 2/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
RAB9A P51151 2/20 0.36
TP53 P04637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20157894 0.92 CES2 (0.50) HTTCES2CES1
SCHEMBL21351893 0.89 RAB9A (0.43) NPC1MAPTSMN1; SMN2RAB9ATP53
SCHEMBL9726681 0.89 CSNK2A1 (0.47) NPC1MAPTMAPK1HTTDGAT1
SCHEMBL27774516 0.89 MAPT (0.44) NPC1MAPTMAPK1HTTCSNK2A1
SCHEMBL20157772 0.86 LOXL2 (0.38) NPC1MAPTMAPK1HTTDGAT1
SCHEMBL20157805 0.86 NPC1 (0.35) NPC1MAPTMAPK1HTTDGAT1
SCHEMBL21550069 0.81 CES2 (0.38) NPC1MAPTMAPK1HTTDGAT1
SCHEMBL20158071 0.81 KMT2A (0.36) NPC1MAPTMAPK1HTTLOXL2
SCHEMBL20157825 0.80 HPGD (0.45) NPC1MAPTHTTCSNK2A1CES2
SCHEMBL11755563 0.80 CES2 (0.50) NPC1MAPTHTTHDAC7CES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086605-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed