SCHEMBL21362762

SCHEMBL21362762

C=Cc1ccc(C(=O)c2ccc(CS(C)(=O)=O)cc2Br)c(Cl)c1

nearest known ligand 0.33

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.33
MCL1 Q07820 3/20 0.32
RCE1 Q9Y256 1/20 0.31
FLT1 P17948 2/20 0.31
FLT4 P35916 2/20 0.31
KDR P35968 2/20 0.31
HPGD P15428 1/20 0.31
ALDH1A1 P00352 1/20 0.31
BCL2L11 O43521 1/20 0.30
BCL2L1 Q07817 1/20 0.30
PTGS2 P35354 1/20 0.30
GRIN1 Q05586 1/20 0.30
KCNH2 Q12809 1/20 0.30
GRIN2B Q13224 1/20 0.30
USP28 Q96RU2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20158005 0.83 HPGD (0.39) PTPN1FLT1FLT4KDRHPGD
SCHEMBL21362178 0.82 NPC1 (0.41) PTPN1FLT1FLT4KDRHPGD
SCHEMBL21362707 0.74 BCL2L11 (0.32) MCL1HPGDBCL2L11BCL2L1PTGS2
SCHEMBL21362746 0.74 TAS1R3 (0.35) MCL1HPGDPTGS2
SCHEMBL21550050 0.73 SMN1; SMN2 (0.42) FLT1FLT4KDRALDH1A1
SCHEMBL20157822 0.72 HPGD (0.38) FLT1FLT4KDRHPGDALDH1A1
SCHEMBL21564804 0.72 CA1 (0.39) HPGD
SCHEMBL20157769 0.71 HPGD (0.39) FLT1FLT4KDRHPGDALDH1A1
SCHEMBL20157951 0.71 MAPT (0.47) PTPN1ALDH1A1
SCHEMBL21564734 0.71 RECQL (0.40) HPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3539960-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF Luoxin Pharmaceutical (Shanghai) Co., Ltd. (CN) 2019-09-18 EP disclosed