SCHEMBL20158037

SCHEMBL20158037

C=C(c1ccc(OC)c(F)c1)c1ccc(CBr)cc1Br

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTT P42858 4/20 0.43
LMNA P02545 2/20 0.43
MAPK1 P28482 1/20 0.43
RAB9A P51151 1/20 0.43
ACHE P22303 1/20 0.43
MEP1B Q16820 1/20 0.38
PDE4A P27815 4/20 0.38
PDE4B Q07343 4/20 0.38
PDE4C Q08493 4/20 0.38
PDE4D Q08499 4/20 0.38
TAS1R3 Q7RTX0 1/20 0.38
TAS1R1 Q7RTX1 1/20 0.38
ALDH1A1 P00352 3/20 0.37
KDM4E B2RXH2 1/20 0.37
MITF O75030 1/20 0.37
TAS2R14 Q9NYV8 1/20 0.36
MEN1 O00255 1/20 0.36
MAPT P10636 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20158040 0.85 ACHE (0.54) HTTLMNAMAPK1RAB9AACHE
SCHEMBL21362429 0.81 SMN1; SMN2 (0.41) RAB9AALDH1A1KDM4EMEN1MAPT
SCHEMBL29442867 0.76 HTT (0.50) HTTLMNAMAPK1RAB9AALDH1A1
SCHEMBL186570 0.76 HTT (0.50) HTTLMNAMAPK1RAB9AALDH1A1
SCHEMBL20157608 0.75 ALDH1A1 (0.44) ACHEALDH1A1TAS2R14
SCHEMBL21362819 0.74 ACHE (0.40) HTTLMNAMAPK1RAB9AACHE
SCHEMBL991185 0.72 HTT (0.56) HTTLMNAMAPK1RAB9AACHE
SCHEMBL20157984 0.72 NPC1 (0.38) HTTLMNARAB9AACHEMEP1B
SCHEMBL29463290 0.71 MAPT (0.56) HTTMAPK1ALDH1A1KDM4EMEN1
SCHEMBL333582 0.71 MAPT (0.56) HTTMAPK1ALDH1A1KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086605-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed