SCHEMBL21362819

SCHEMBL21362819

COc1cc(C(=O)c2ccc(CBr)cc2Br)c(C)cc1F

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.40
LCK P06239 1/20 0.38
FYN P06241 1/20 0.38
ALDH1A1 P00352 2/20 0.38
HTT P42858 3/20 0.37
RAB9A P51151 2/20 0.37
LMNA P02545 2/20 0.37
MAPK1 P28482 1/20 0.37
KDM4E B2RXH2 1/20 0.36
MITF O75030 1/20 0.36
POLB P06746 1/20 0.36
KMT2A Q03164 1/20 0.36
NPC1 O15118 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MEP1B Q16820 1/20 0.35
CYP4F2 P78329 1/20 0.35
CYP4A11 Q02928 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20157984 0.88 NPC1 (0.38) ACHELCKFYNALDH1A1HTT
SCHEMBL20158038 0.87 CYP4F2 (0.40) ACHELCKFYNALDH1A1HTT
SCHEMBL21362528 0.85 LCK (0.42) LCKFYNALDH1A1HTTRAB9A
SCHEMBL20157608 0.84 ALDH1A1 (0.44) ACHEALDH1A1
SCHEMBL20158040 0.84 ACHE (0.54) ACHEALDH1A1HTTRAB9ALMNA
SCHEMBL20157512 0.81 NPC1 (0.46) LCKFYNALDH1A1RAB9AKMT2A
SCHEMBL20157609 0.80 ALDH1A1 (0.46) ACHEALDH1A1KMT2ANPC1
SCHEMBL20158023 0.80 ABL1 (0.45) ACHELCKFYNALDH1A1HTT
SCHEMBL21564879 0.77 CYP4F2 (0.37) ALDH1A1LMNAKDM4EMEP1BCYP4F2
SCHEMBL20157772 0.77 LOXL2 (0.38) ALDH1A1HTTLMNAMAPK1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3539960-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF Luoxin Pharmaceutical (Shanghai) Co., Ltd. (CN) 2019-09-18 EP disclosed