SCHEMBL2015807

SCHEMBL2015807

OCCc1ccc2cccnc2c1-c1cncc(F)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 1/20 0.36
KDM4E B2RXH2 5/20 0.36
NPC1 O15118 4/20 0.36
RAB9A P51151 4/20 0.36
L3MBTL1 Q9Y468 3/20 0.36
CCR1 P32246 2/20 0.36
CCR5 P51681 2/20 0.36
CCR8 P51685 2/20 0.36
CYP3A4 P08684 2/20 0.36
GMNN O75496 1/20 0.36
LMNA P02545 1/20 0.36
TP53 P04637 1/20 0.36
HSP90AA1 P07900 1/20 0.36
MMP2 P08253 1/20 0.36
CYP2D6 P10635 1/20 0.36
MAPT P10636 1/20 0.36
MMP9 P14780 1/20 0.36
ALOX15 P16050 1/20 0.36
TSHR P16473 1/20 0.36
NFKB1 P19838 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2013343 0.88 KDM4E (0.36) KDM4ENPC1RAB9AL3MBTL1CCR1
SCHEMBL2011511 0.87 KDM4E (0.40) MAPK14KDM4ENPC1RAB9AL3MBTL1
SCHEMBL2012265 0.85 PIK3CD (0.42) KDM4ENPC1RAB9ACCR1CCR5
SCHEMBL2718191 0.77 KDM4E (0.42) KDM4ENPC1RAB9AL3MBTL1CCR1
SCHEMBL2015805 0.76 PIK3CD (0.43) KDM4ENPC1RAB9AL3MBTL1CCR1
SCHEMBL2050742 0.75 PIK3CD (0.42) KDM4ENPC1RAB9AL3MBTL1CYP3A4
SCHEMBL2010932 0.74 KDM4E (0.43) KDM4ENPC1RAB9AL3MBTL1CCR1
SCHEMBL2011836 0.74 LMNA (0.40) KDM4ENPC1RAB9ACCR1CCR5
SCHEMBL2013339 0.73 PIK3CD (0.43) KDM4ECCR1CCR5CCR8CYP3A4
SCHEMBL2011259 0.72 TAAR1 (0.43) KDM4ENPC1RAB9ACCR1CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011075630-A1 SUBSTITUTED FUSED ARYL AND HETEROARYL DERIVATIVES AS PI3K INHIBITORS INCYTE CORPORATION (US) 2011-06-23 WO disclosed