SCHEMBL2010932

SCHEMBL2010932

OCCc1ccc2cccnc2c1-c1ccccc1F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.43
LMNA P02545 4/20 0.43
MAPT P10636 3/20 0.43
HTT P42858 2/20 0.43
TDP1 Q9NUW8 2/20 0.43
TP53 P04637 2/20 0.43
MMP2 P08253 2/20 0.43
TSHR P16473 2/20 0.43
GMNN O75496 1/20 0.43
HSP90AA1 P07900 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
MMP9 P14780 1/20 0.43
ALOX15 P16050 1/20 0.43
NFKB1 P19838 1/20 0.43
MMP8 P22894 1/20 0.43
CCR1 P32246 1/20 0.43
THPO P40225 1/20 0.43
MTOR P42345 1/20 0.43
MMP13 P45452 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2016907 0.88 KDM4E (0.44) KDM4ELMNAMAPTHTTTDP1
SCHEMBL2014257 0.80 KDM4E (0.42) KDM4ELMNAMAPTHTTTDP1
SCHEMBL2011511 0.78 KDM4E (0.40) KDM4ELMNAMAPTHTTTDP1
SCHEMBL2015203 0.77 CDK1 (0.46) KDM4ELMNAMAPTHTTTDP1
SCHEMBL2012265 0.76 PIK3CD (0.42) KDM4ELMNAMAPTHTTTDP1
SCHEMBL2015807 0.74 MAPK14 (0.36) KDM4ELMNAMAPTHTTTDP1
SCHEMBL2010930 0.73 TP53 (0.44) KDM4ELMNAMAPTHTTTDP1
SCHEMBL2014256 0.73 ALDH1A1 (0.44) KDM4ELMNAMAPTHTTTDP1
SCHEMBL30203803 0.71 HDAC6 (0.52) KDM4ELMNAMAPTHTTTDP1
SCHEMBL11497495 0.71 HDAC6 (0.52) KDM4ELMNAMAPTHTTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011075630-A1 SUBSTITUTED FUSED ARYL AND HETEROARYL DERIVATIVES AS PI3K INHIBITORS INCYTE CORPORATION (US) 2011-06-23 WO disclosed