SCHEMBL20158083

SCHEMBL20158083

Cc1ccc(C(O)c2ccc([C@@H](C)O)c(F)c2)c(Br)c1

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.34
LMNA P02545 1/20 0.34
CHRM1 P11229 1/20 0.34
SLC6A2 P23975 1/20 0.34
ADRA1A P35348 1/20 0.34
HTR2B P41595 1/20 0.34
PDE2A O00408 3/20 0.33
AKR1C3 P42330 1/20 0.32
AKR1C2 P52895 1/20 0.32
PTGS2 P35354 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20157992 0.82 TOP2A (0.40) LMNA
SCHEMBL21362648 0.81 ACHE (0.39) TRPA1LMNACHRM1SLC6A2ADRA1A
SCHEMBL20157895 0.79 TOP2A (0.37) LMNA
SCHEMBL2474757 0.79 LMNA (0.47) TRPA1LMNACHRM1SLC6A2ADRA1A
SCHEMBL28493300 0.79 LMNA (0.47) TRPA1LMNACHRM1SLC6A2ADRA1A
SCHEMBL13345087 0.79 TRPA1 (0.47) TRPA1LMNACHRM1SLC6A2ADRA1A
SCHEMBL21564876 0.75 LMNA (0.34) TRPA1LMNACHRM1SLC6A2ADRA1A
SCHEMBL11859495 0.74 MLKL (0.45) TRPA1LMNACHRM1SLC6A2ADRA1A
SCHEMBL21550255 0.74 TRPA1 (0.33) TRPA1LMNACHRM1SLC6A2ADRA1A
SCHEMBL20157481 0.72 TOP2A (0.39) LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086605-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed