SCHEMBL20159137

SCHEMBL20159137

C[C@H]1CN(c2cccc3ccn(COCC[Si](C)(C)C)c23)CCN1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.34
CREBBP Q92793 1/20 0.34
HTR2C P28335 1/20 0.32
KHK P50053 2/20 0.32
MKNK1 Q9BUB5 2/20 0.32
MKNK2 Q9HBH9 2/20 0.32
CDK1 P06493 1/20 0.32
CDK2 P24941 1/20 0.32
PRKCQ Q04759 3/20 0.32
PRKCD Q05655 1/20 0.32
ROCK2 O75116 1/20 0.32
FLT3 P36888 1/20 0.32
CAMK2D Q13557 1/20 0.32
PIM2 Q9P1W9 1/20 0.32
WEE1 P30291 1/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
CHEK1 O14757 2/20 0.31
MLNR O43193 1/20 0.31
PDE5A O76074 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20142084 0.76 MAP4K4 (0.41)
SCHEMBL4503124 0.72 ADRA2A (0.43) DGAT1KLKB1
SCHEMBL6030125 0.71 DGAT1 (0.40) LMNADGAT1
SCHEMBL30018075 0.71 DGAT1 (0.38) HTR2CDGAT1
SCHEMBL15823309 0.69 DGAT1 (0.34) HTR2CDGAT1
SCHEMBL20142085 0.69 KLKB1 (0.30) DGAT1KLKB1
SCHEMBL15824847 0.69 DGAT1 (0.34) DGAT1
SCHEMBL20140653 0.67 PIM1 (0.41) HTR2CKHKMKNK1MKNK2CDK1
SCHEMBL20140655 0.67 PIM1 (0.41) HTR2CKHKMKNK1MKNK2CDK1
SCHEMBL1258087 0.66 CDK4 (0.49) HTR2CFLT3ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089493-A1 PYRROLE mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed