SCHEMBL20159647

SCHEMBL20159647

NC1C2CC1N(c1ccnc(Cl)c1)C2

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 9/20 0.40
CHRNB4 P30926 9/20 0.40
CHRNA3 P32297 9/20 0.40
CHRNA4 P43681 9/20 0.40
CYP17A1 P05093 4/20 0.37
CHRM1 P11229 1/20 0.34
LOX P28300 1/20 0.34
LOXL3 P58215 1/20 0.34
LOXL2 Q9Y4K0 1/20 0.34
HCRTR1 O43613 1/20 0.32
HCRTR2 O43614 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20159687 0.78 NR1H2 (0.41) CHRNB2CHRNB4CHRNA3CHRNA4CYP17A1
SCHEMBL20159656 0.78 CHRNA3 (0.39) CHRNB2CHRNB4CHRNA3CHRNA4CYP17A1
SCHEMBL23504817 0.78 HCRTR1 (0.44) CHRNB2CHRNB4CHRNA3CHRNA4HCRTR1
SCHEMBL23504791 0.76 MMP2 (0.32) CHRNB2CHRNB4CHRNA3CHRNA4CYP17A1
SCHEMBL18970901 0.74 CHRM4 (0.38) CHRNB2CHRNB4CHRNA3CHRNA4CYP17A1
SCHEMBL20609193 0.74 CHRM4 (0.38) CHRNB2CHRNB4CHRNA3CHRNA4CYP17A1
SCHEMBL20031740 0.74 CHRM4 (0.38) CHRNB2CHRNB4CHRNA3CHRNA4CYP17A1
SCHEMBL20609194 0.74 CHRM4 (0.38) CHRNB2CHRNB4CHRNA3CHRNA4CYP17A1
SCHEMBL18952559 0.74 CHRM4 (0.38) CHRNB2CHRNB4CHRNA3CHRNA4CYP17A1
SCHEMBL20159356 0.72 CHRM4 (0.32) CYP17A1LOXLOXL3LOXL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018087018-A1 PHENOXYTRIAZOLES F. HOFFMANN-LA ROCHE AG (CH) 2018-05-17 WO disclosed