SCHEMBL20159982

SCHEMBL20159982

CC(C)n1nc(N)nc1Oc1ccc(F)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN4A P35499 3/20 0.38
L3MBTL1 Q9Y468 1/20 0.37
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
SCN9A Q15858 4/20 0.36
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
RET P07949 1/20 0.34
HTT P42858 1/20 0.34
NCOA3 Q9Y6Q9 1/20 0.34
KCNH2 Q12809 2/20 0.34
SCN5A Q14524 2/20 0.34
HTR7 P34969 3/20 0.33
ADRA1D P25100 1/20 0.33
ADRA1A P35348 1/20 0.33
ADRA1B P35368 1/20 0.33
PIK3CD O00329 1/20 0.33
ABL1 P00519 1/20 0.33
EGFR P00533 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20159730 0.83 MAP4K4 (0.39) KDM4EALDH1A1MAPTPIK3CDABL1
SCHEMBL20138803 0.82 SCN4A (0.38) SCN4AL3MBTL1MEN1KMT2ASCN9A
SCHEMBL20159299 0.79 HTR2A (0.37) KDM4EALDH1A1MAPTKCNH2PIK3CD
SCHEMBL20159650 0.74 PSEN1 (0.51) SCN9ASCN5AHTR7ABL1SRC
SCHEMBL10793571 0.70 MPO (0.39) MEN1KMT2AKCNH2PIK3CDABL1
SCHEMBL23504771 0.67 HTR2A (0.41) L3MBTL1SCN9A
SCHEMBL20138669 0.67 HTR2A (0.41) L3MBTL1SCN9AKCNH2SCN5A
SCHEMBL20142954 0.67 MAP4K4 (0.35) L3MBTL1ALDH1A1MAPTHTTPIK3CD
SCHEMBL20138683 0.67
SCHEMBL20142991 0.67 MAPT (0.37) KDM4EMEN1KMT2ASCN9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018087018-A1 PHENOXYTRIAZOLES F. HOFFMANN-LA ROCHE AG (CH) 2018-05-17 WO disclosed