SCHEMBL20160027

SCHEMBL20160027

Cc1nnc2c(C(N)=O)cc(Cl)nn12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.40
RXFP1 Q9HBX9 1/20 0.40
NNMT P40261 2/20 0.36
BRD9 Q9H8M2 1/20 0.35
PDE4B Q07343 2/20 0.34
PIK3CD O00329 1/20 0.34
ABL1 P00519 1/20 0.34
EGFR P00533 1/20 0.34
HCK P08631 1/20 0.34
SRC P12931 1/20 0.34
KDR P35968 1/20 0.34
PIK3CA P42336 1/20 0.34
PIK3CB P42338 1/20 0.34
MTOR P42345 1/20 0.34
EPHB4 P54760 1/20 0.34
PRKDC P78527 1/20 0.34
PI4KB Q9UBF8 1/20 0.34
PDE4A P27815 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14246825 0.86 L3MBTL1 (0.41) L3MBTL1RXFP1BRD9BRD4TSHR
SCHEMBL20160352 0.84 CYP1A2 (0.36) L3MBTL1RXFP1NNMTBRD9BRD4
SCHEMBL20160235 0.83 NNMT (0.34) L3MBTL1RXFP1NNMTBRD9PDE4B
SCHEMBL16140295 0.82 RXFP1 (0.38) L3MBTL1RXFP1BRD9BRD4CREBBP
SCHEMBL16244413 0.75 RXFP1 (0.45) L3MBTL1RXFP1BRD9BRD4CREBBP
SCHEMBL15711661 0.74 RXFP1 (0.47) L3MBTL1RXFP1BRD9BRD4CREBBP
SCHEMBL16244643 0.74 BRD9 (0.50) L3MBTL1RXFP1BRD9BRD4CREBBP
SCHEMBL6620694 0.72 RXFP1 (0.42) L3MBTL1RXFP1BRD9BRD4CREBBP
SCHEMBL16244397 0.72 RXFP1 (0.37) L3MBTL1RXFP1BRD9BRD4CREBBP
SCHEMBL11283623 0.70 CASP1 (0.33) NNMTSYKCASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086585-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed