SCHEMBL20160352

SCHEMBL20160352

Cc1cc(C(N)=O)c2nnc(C)n2n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.36
AURKA O14965 1/20 0.36
CSF1R P07333 1/20 0.36
RET P07949 1/20 0.36
LTK P29376 1/20 0.36
CSNK1A1 P48729 1/20 0.36
CDK8 P49336 1/20 0.36
CLK2 P49760 1/20 0.36
CDK5 Q00535 1/20 0.36
ACVR1 Q04771 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36
LMNA P02545 1/20 0.36
L3MBTL1 Q9Y468 2/20 0.35
NNMT P40261 2/20 0.35
RXFP1 Q9HBX9 1/20 0.35
BRD9 Q9H8M2 1/20 0.34
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33
HSD17B10 Q99714 1/20 0.33
RCE1 Q9Y256 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20160235 0.85 NNMT (0.34) AURKACSF1RRETLTKCSNK1A1
SCHEMBL20160027 0.84 L3MBTL1 (0.40) ACVR1L3MBTL1NNMTRXFP1BRD9
SCHEMBL20159899 0.73 RXFP1 (0.40) LMNAL3MBTL1RXFP1BRD9TSHR
SCHEMBL16259900 0.71 ALDH1A1 (0.46) CYP1A2LMNARXFP1BRD9BRD4
SCHEMBL14246870 0.71 KAT2A (0.40) L3MBTL1RXFP1BRD9TSHRMAPK1
SCHEMBL14246871 0.71 KAT2A (0.40) L3MBTL1RXFP1BRD9TSHRMAPK1
SCHEMBL25151509 0.70 LMNA (0.49) LMNAL3MBTL1NNMTHSD17B10RCE1
SCHEMBL16556413 0.67 BRD4 (0.51) LMNAL3MBTL1RXFP1BRD9TSHR
SCHEMBL16140295 0.66 RXFP1 (0.38) LMNAL3MBTL1RXFP1BRD9TSHR
SCHEMBL3284181 0.66 CYP1A2 (0.74) CYP1A2LMNANNMTRXFP1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086585-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed