SCHEMBL20160404

SCHEMBL20160404

CCC(=O)C(=O)Cc1ccc(Oc2ccc(F)cc2F)c(I)c1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 2/20 0.39
FAAH O00519 1/20 0.38
HSPB1 P04792 3/20 0.38
CARM1 Q86X55 2/20 0.37
PRMT6 Q96LA8 2/20 0.37
BRD4 O60885 2/20 0.36
NR3C1 P04150 1/20 0.36
NR1I2 O75469 1/20 0.36
PPARG P37231 1/20 0.36
AGTR2 P50052 1/20 0.36
MEN1 O00255 1/20 0.36
BLM P54132 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20160339 0.77 BRD4 (0.52) TRPA1BRD4
SCHEMBL30498824 0.70 PTGS2 (0.56) BRD4
SCHEMBL15067969 0.70 PTGS2 (0.56) BRD4
SCHEMBL28641777 0.70 GAA (0.53) NR1I2PPARGAGTR2MEN1BLM
SCHEMBL20159992 0.68 BRD4 (0.57) BRD4
SCHEMBL30159449 0.68 TRPA1 (0.53) TRPA1HSPB1
SCHEMBL15068172 0.68 EPAS1 (0.52) HSPB1BRD4
SCHEMBL21904840 0.68 HSPB1 (0.72) HSPB1MEN1KMT2A
SCHEMBL25191080 0.68 TRPA1 (0.45) TRPA1HSPB1BRD4
SCHEMBL10456772 0.67 TRPA1 (0.56) TRPA1HSPB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086585-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed