SCHEMBL20160880

SCHEMBL20160880

Cc1cc(C)c(CN)c(OCc2ccccc2)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.48
TSHR P16473 2/20 0.45
AOC3 Q16853 1/20 0.45
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
HTT P42858 2/20 0.41
STAT3 P40763 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
ATP4A P20648 1/20 0.41
ATP4B P51164 1/20 0.41
MAOB P27338 1/20 0.41
ALDH1A1 P00352 2/20 0.40
LMNA P02545 3/20 0.40
POLB P06746 2/20 0.40
RAB9A P51151 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
OPRM1 P35372 1/20 0.40
OPRK1 P41145 1/20 0.40
CDK1 P06493 1/20 0.40
CCNB1 P14635 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30535930 0.85 L3MBTL1 (0.48) L3MBTL1TSHRMEN1KMT2AHTT
SCHEMBL15814340 0.85 L3MBTL1 (0.48) L3MBTL1TSHRMEN1KMT2AHTT
SCHEMBL29779070 0.85 L3MBTL1 (0.48) L3MBTL1TSHRMEN1KMT2AHTT
SCHEMBL15814471 0.85 L3MBTL1 (0.48) L3MBTL1TSHRMEN1KMT2AHTT
SCHEMBL20160832 0.85 TSHR (0.48) L3MBTL1TSHRAOC3MEN1KMT2A
SCHEMBL18526223 0.81 MEN1 (0.46) L3MBTL1TSHRAOC3MEN1KMT2A
SCHEMBL21419430 0.80 AOC3 (0.41) L3MBTL1TSHRAOC3MEN1KMT2A
SCHEMBL17874237 0.79 AOC3 (0.41) L3MBTL1TSHRAOC3HTTSTAT3
SCHEMBL18526460 0.79 L3MBTL1 (0.42) L3MBTL1TSHRMEN1KMT2AHTT
SCHEMBL15813749 0.79 USP28 (0.47) L3MBTL1MEN1KMT2AHTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086589-A1 1,5,7-TRI-SUBSTITUTED ISOQUINOLINE DERIVATIVES, PREPARATION THEREOF, AND USE THEREOF IN MEDICINES 上海海雁医药科技有限公司 2018-05-17 WO disclosed