SCHEMBL20160832

SCHEMBL20160832

CCc1cc(C)nc(OCc2ccccc2)c1CN

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.48
AOC3 Q16853 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.44
MGMT P16455 2/20 0.40
CDK1 P06493 1/20 0.40
CCNB1 P14635 1/20 0.40
CCNA2 P20248 1/20 0.40
CDK2 P24941 1/20 0.40
CCNA1 P78396 1/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
ATP4A P20648 1/20 0.39
ATP4B P51164 1/20 0.39
STAT3 P40763 1/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HCAR2 Q8TDS4 1/20 0.39
MEN1 O00255 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15814133 0.86 TSHR (0.45) TSHRL3MBTL1MGMTCDK1CCNB1
SCHEMBL15815024 0.86 TSHR (0.45) TSHRL3MBTL1MGMTCDK1CCNB1
SCHEMBL20160880 0.85 L3MBTL1 (0.48) TSHRAOC3L3MBTL1MGMTCDK1
SCHEMBL15814853 0.80 TSHR (0.46) TSHRL3MBTL1MGMTCDK1CCNB1
SCHEMBL18526223 0.78 MEN1 (0.46) TSHRAOC3L3MBTL1ATP4AATP4B
SCHEMBL18526569 0.78 AOC3 (0.43) TSHRAOC3L3MBTL1ATP4AATP4B
SCHEMBL15814214 0.77 SQOR (0.55) TSHRL3MBTL1HTTSMN1; SMN2ALDH1A1
SCHEMBL21419430 0.77 AOC3 (0.41) TSHRAOC3L3MBTL1ATP4AATP4B
SCHEMBL30466417 0.76 L3MBTL1 (0.43) TSHRL3MBTL1STAT3HTTSMN1; SMN2
SCHEMBL17874237 0.76 AOC3 (0.41) TSHRAOC3L3MBTL1ATP4AATP4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086589-A1 1,5,7-TRI-SUBSTITUTED ISOQUINOLINE DERIVATIVES, PREPARATION THEREOF, AND USE THEREOF IN MEDICINES 上海海雁医药科技有限公司 2018-05-17 WO disclosed