SCHEMBL2016172

SCHEMBL2016172

O=C(O)Nc1cnc(Cl)c(F)c1I

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.33
NPC1 O15118 1/20 0.33
NTRK1 P04629 2/20 0.33
BRD4 O60885 1/20 0.33
RAB9A P51151 1/20 0.31
POLB P06746 1/20 0.31
P4HTM Q9NXG6 2/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19950148 0.81 NPC1 (0.34) SMN1; SMN2NPC1NTRK1BRD4RAB9A
SCHEMBL30038835 0.78 ATR (0.42)
SCHEMBL2019695 0.78 ATR (0.42)
SCHEMBL21773064 0.78 XPO1 (0.35) SMN1; SMN2NPC1NTRK1RAB9A
SCHEMBL26697648 0.78 POLB (0.36) BRD4POLB
SCHEMBL26697721 0.76 ALDH1A1 (0.35) SMN1; SMN2NPC1NTRK1BRD4RAB9A
SCHEMBL12395995 0.75
SCHEMBL26988407 0.75 BRD4 (0.35) SMN1; SMN2NPC1NTRK1BRD4RAB9A
SCHEMBL25337174 0.74 KEAP1 (0.42) SMN1; SMN2NPC1RAB9A
SCHEMBL16165254 0.72 RAB9A (0.41) SMN1; SMN2NPC1BRD4RAB9APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3740478-B1 FUSED IMIDAZOLE DERIVATIVES AS IL-17 MODULATORS UCB Biopharma SRL (BE) 2023-11-01 EP disclosed
US-11472794-B2 Fused imidazole derivatives as IL-17 modulators UCB Biopharma SRL (BE) 2022-10-18 US disclosed
EP-3844158-A1 HETEROARYL-SUBSTITUTED SULFONAMIDE COMPOUNDS AND THEIR USE AS SODIUM CHANNEL INHIBITORS Xenon Pharmaceuticals Inc. (CA) 2021-07-07 EP disclosed
US-20210053952-A1 Fused Imidazole Derivatives as IL-17 Modulators UCB Biopharma SRL (BE) 2021-02-25 US disclosed
EP-3740478-A1 FUSED IMIDAZOLE DERIVATIVES AS IL-17 MODULATORS UCB Biopharma SRL (BE) 2020-11-25 EP disclosed
US-10752623-B2 Heteroaryl-substituted sulfonamide compounds and their use as sodium channel inhibitors XENON PHARMACEUTICALS INC. (CA) 2020-08-25 US disclosed
WO-2020047312-A1 HETEROARYL-SUBSTITUTED SULFONAMIDE COMPOUNDS AND THEIR USE AS SODIUM CHANNEL INHIBITORS XENON PHARMACEUTICALS INC. (CA) 2020-03-05 WO disclosed
US-20200071313-A1 HETEROARYL-SUBSTITUTED SULFONAMIDE COMPOUNDS AND THEIR USE AS SODIUM CHANNEL INHIBITORS XENON PHARMACEUTICALS INC. (CA) 2020-03-05 US disclosed
EP-2513110-A1 1, 7 - DIAZACARBAZOLES AND THEIR USE IN THE TREATMENT OF CANCER F. Hoffmann-La Roche AG (CH) 2012-10-24 EP disclosed
WO-2011073263-A1 1, 7 - DIAZACARBAZOLES AND THEIR USE IN THE TREATMENT OF CANCER F. HOFFMANN-LA ROCHE AG (CH) 2011-06-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200071313-A1 HETEROARYL-SUBSTITUTED SULFONAMIDE COMPOUNDS AND THEIR USE AS SODIUM CHANNEL INHIBITORS SCN1A, SCN2A, SCN2B SMN1; SMN2 331/4885NPC1 659/4885NTRK1 888/4885
US-11472794-B2 Fused imidazole derivatives as IL-17 modulators IL17A, IL2, IL23R SMN1; SMN2 4168/4885NPC1 3094/4885NTRK1 1510/4885
US-10752623-B2 Heteroaryl-substituted sulfonamide compounds and their use as sodium channel inhibitors SCN1A, SCN2A, SCN2B SMN1; SMN2 331/4885NPC1 659/4885NTRK1 888/4885
US-20210053952-A1 Fused Imidazole Derivatives as IL-17 Modulators IL17A, IL2, IL23R SMN1; SMN2 4168/4885NPC1 3094/4885NTRK1 1510/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.