SCHEMBL19950148

SCHEMBL19950148

Cc1c(NC(=O)O)cnc(Cl)c1F

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.34
SMN1; SMN2 Q16637 4/20 0.34
NTRK1 P04629 2/20 0.33
BRD4 O60885 1/20 0.33
KCNQ3 O43525 2/20 0.33
KCNQ2 O43526 2/20 0.33
KCNE1 P15382 2/20 0.33
KCNQ1 P51787 2/20 0.33
KCNQ5 Q9NR82 1/20 0.33
RAB9A P51151 4/20 0.33
ALDH1A1 P00352 2/20 0.33
GAA P10253 2/20 0.33
DHODH Q02127 1/20 0.32
KMT2A Q03164 1/20 0.32
GPR35 Q9HC97 1/20 0.32
PIK3C3 Q8NEB9 1/20 0.32
GRM5 P41594 1/20 0.32
KDM4E B2RXH2 1/20 0.31
TP53 P04637 1/20 0.31
GLA P06280 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2016172 0.81 SMN1; SMN2 (0.33) NPC1SMN1; SMN2NTRK1BRD4RAB9A
SCHEMBL26988407 0.80 BRD4 (0.35) NPC1SMN1; SMN2NTRK1BRD4KCNQ3
SCHEMBL21773064 0.79 XPO1 (0.35) NPC1SMN1; SMN2NTRK1KCNQ3KCNQ2
SCHEMBL26697648 0.79 POLB (0.36) BRD4ALDH1A1KMT2APOLB
SCHEMBL26697721 0.78 ALDH1A1 (0.35) NPC1SMN1; SMN2NTRK1BRD4KCNQ3
SCHEMBL19950247 0.77 MEN1 (0.36) NPC1SMN1; SMN2RAB9AALDH1A1KMT2A
SCHEMBL27185426 0.75 KEAP1 (0.42) NPC1SMN1; SMN2RAB9AALDH1A1DHODH
SCHEMBL15204699 0.74 AGBL2 (0.40) NPC1SMN1; SMN2KCNQ3KCNQ2KCNE1
SCHEMBL16165254 0.74 RAB9A (0.41) NPC1SMN1; SMN2BRD4RAB9AALDH1A1
SCHEMBL30388447 0.71 SMN1; SMN2 (0.39) NPC1SMN1; SMN2RAB9AALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240034736-A1 HSD17B13 INHIBITORS AND USES THEREOF FL2022-001, INC. 2024-02-01 US disclosed
US-11795166-B2 Pyrazolopyridine compounds and uses thereof INCYTE CORPORATION (US) 2023-10-24 US disclosed
EP-4221702-A1 HSD17B13 INHIBITORS AND USES THEREOF FL2022-001, Inc. (US) 2023-08-09 EP disclosed
EP-4119558-A1 PYRAZOLOPYRIDINE COMPOUNDS AND USES THEREOF Incyte Corporation (US) 2023-01-18 EP disclosed
EP-3510032-B1 PYRAZOLOPYRIDINE DERIVATIVES AS HPK1 MODULATORS AND USES THEREOF FOR THE TREATMENT OF CANCER INCYTE CORP (US) 2022-07-06 EP disclosed
US-20210380581-A1 PYRAZOLOPYRIDINE COMPOUNDS AND USES THEREOF INCYTE CORPORATION 2021-12-09 US disclosed
US-10934288-B2 Pyrazolopyridine compounds and uses thereof INCYTE CORPORATION (US) 2021-03-02 US disclosed
US-20200087301-A1 PYRAZOLOPYRIDINE COMPOUNDS AND USES THEREOF INCYTE CORPORATION 2020-03-19 US disclosed
US-10435405-B2 Pyrazolopyridine compounds and uses thereof INCYTE CORPORATION (US) 2019-10-08 US disclosed
EP-3510032-A1 PYRAZOLOPYRIDINE DERIVATIVES AS HPK1 MODULATORS AND USES THEREOF FOR THE TREATMENT OF CANCER Incyte Corporation (US) 2019-07-17 EP disclosed
US-10266530-B2 Pyrazolopyridine compounds and uses thereof INCYTE CORPORATION (US) 2019-04-23 US disclosed
US-20190106419-A1 PYRAZOLOPYRIDINE COMPOUNDS AND USES THEREOF INCYTE CORPORATION 2019-04-11 US disclosed
WO-2018049200-A1 PYRAZOLOPYRIDINE DERIVATIVES AS HPK1 MODULATORS AND USES THEREOF FOR THE TREATMENT OF CANCER INCYTE CORPORATION (US) 2018-03-15 WO disclosed
US-20180072720-A1 PYRAZOLOPYRIDINE COMPOUNDS AND USES THEREOF INCYTE CORPORATION 2018-03-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200087301-A1 PYRAZOLOPYRIDINE COMPOUNDS AND USES THEREOF PDXK, PCK1, PGK1 NPC1 754/4885SMN1; SMN2 3405/4885NTRK1 2377/4885
US-11795166-B2 Pyrazolopyridine compounds and uses thereof PDXK, PCK1, PGK1 NPC1 754/4885SMN1; SMN2 3405/4885NTRK1 2377/4885
US-20180072720-A1 PYRAZOLOPYRIDINE COMPOUNDS AND USES THEREOF PDXK, PCK1, PGK1 NPC1 754/4885SMN1; SMN2 3405/4885NTRK1 2377/4885
US-10934288-B2 Pyrazolopyridine compounds and uses thereof PDXK, PCK1, PGK1 NPC1 754/4885SMN1; SMN2 3405/4885NTRK1 2377/4885
US-20210380581-A1 PYRAZOLOPYRIDINE COMPOUNDS AND USES THEREOF PDXK, PCK1, PGK1 NPC1 754/4885SMN1; SMN2 3405/4885NTRK1 2377/4885
US-20240034736-A1 HSD17B13 INHIBITORS AND USES THEREOF HSD17B3, HSD17B11, HSD17B1 NPC1 332/4885SMN1; SMN2 3176/4885NTRK1 4805/4885
US-10435405-B2 Pyrazolopyridine compounds and uses thereof PDXK, PCK1, PGK1 NPC1 754/4885SMN1; SMN2 3405/4885NTRK1 2377/4885
US-20190106419-A1 PYRAZOLOPYRIDINE COMPOUNDS AND USES THEREOF PDXK, PCK1, PGK1 NPC1 754/4885SMN1; SMN2 3405/4885NTRK1 2377/4885
US-10266530-B2 Pyrazolopyridine compounds and uses thereof PDXK, PCK1, PGK1 NPC1 754/4885SMN1; SMN2 3405/4885NTRK1 2377/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.