SCHEMBL20161748

SCHEMBL20161748

CC(C)N1[C@@H]2CC[C@H]1CN(C)C2

nearest known ligand 0.33

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.33
CYP2C9 P11712 1/20 0.33
OPRM1 P35372 1/20 0.32
HSD11B1 P28845 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7848572 1.00 LMNA (0.33) LMNACYP2C9OPRM1HSD11B1
SCHEMBL13791826 0.90 MAPK1 (0.37)
SCHEMBL19763596 0.86 NCF1 (0.32)
SCHEMBL20071156 0.84
SCHEMBL27280941 0.80 LMNA (0.31) LMNACYP2C9OPRM1
SCHEMBL761435 0.80 LMNA (0.35) LMNACYP2C9
SCHEMBL9963382 0.80 LMNA (0.35) LMNACYP2C9
SCHEMBL24816724 0.79 HRH3 (0.30)
SCHEMBL9884491 0.79 HRH3 (0.30)
SCHEMBL12267691 0.79 HRH3 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11807636-B2 IRAK degraders and uses thereof KYMERA THERAPEUTICS, INC. (US) 2023-11-07 US disclosed
WO-2023192586-A1 IRAK DEGRADERS AND USES THEREOF KYMERA THERAPEUTICS, INC. (US) 2023-10-05 WO disclosed
US-20230183216-A1 PYRIDIZIN-3(2H)-ONE DERIVATIVES GILEAD SCIENCES, INC. 2023-06-15 US disclosed
WO-2023098656-A1 COMPOUNDS FOR THE DEGRADATION OF EGFR KINASE BEIGENE, LTD. (GB) 2023-06-08 WO disclosed
WO-2022189810-A1 ANTI-VIRAL COMPOUNDS Infex Therapeutics Limited (GB) 2022-09-15 WO disclosed
US-11358949-B2 Carbamate and urea compounds as multikinase inhibitors ANGEX PHARMACEUTICAL, INC. (US) 2022-06-14 US disclosed
US-20210163445-A1 CARBAMATE AND UREA COMPOUNDS AS MULTIKINASE INHIBITORS ANGEX PHARMACEUTICAL, INC. 2021-06-03 US disclosed
US-11008314-B2 Compounds and methods for modulating interleukin-2-inducible t-cell kinase CORVUS PHARMACEUTICALS, INC. (US) 2021-05-18 US disclosed
WO-2020108613-A1 HETEROAROMATIC DERIVATIVES FOR USE AS REGULATOR, PREPARATION METHOD THEREFOR AND USE THEREOF 江苏豪森药业集团有限公司 2020-06-04 WO disclosed
WO-2018089261-A2 COMPOUNDS AND METHODS FOR MODULATING INTERLEUKIN-2-INDUCIBLE T-CELL KINASE CORVUS PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11008314-B2 Compounds and methods for modulating interleukin-2-inducible t-cell kinase IL2, NFATC1, IL2RA LMNA 4243/4885CYP2C9 4795/4885OPRM1 4350/4885
US-11807636-B2 IRAK degraders and uses thereof IRAK2, IRAK3, IRAK1 LMNA 1656/4885CYP2C9 3608/4885OPRM1 4472/4885
US-20230183216-A1 PYRIDIZIN-3(2H)-ONE DERIVATIVES PIR, CYP3A43, CYP1A2 LMNA 678/4885CYP2C9 168/4885OPRM1 549/4885
US-11358949-B2 Carbamate and urea compounds as multikinase inhibitors UCK2, ULK2, CDK9 LMNA 3217/4885CYP2C9 1950/4885OPRM1 4192/4885
US-20210163445-A1 CARBAMATE AND UREA COMPOUNDS AS MULTIKINASE INHIBITORS UCK2, ULK2, CDK9 LMNA 3217/4885CYP2C9 1950/4885OPRM1 4192/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.